Compile Data Set for Download or QSAR
maximum 50k data
Found 64 with Last Name = 'logan' and Initial = 'me'
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009228(CHEMBL413846 | SP (substance P) | Spantide)
Affinity DataIC50:  0.120nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002373(1-(1-ethynyl)-15a,17a-dimethyl-(1R,15aS,17aS)-2,3,...)
Affinity DataIC50:  24nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002373(1-(1-ethynyl)-15a,17a-dimethyl-(1R,15aS,17aS)-2,3,...)
Affinity DataIC50:  48nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002373(1-(1-ethynyl)-15a,17a-dimethyl-(1R,15aS,17aS)-2,3,...)
Affinity DataIC50:  50nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002384(15a,17a-dimethyl-1-vinyl-(1R,15aS,17aS)-2,3,3a,3b,...)
Affinity DataIC50:  86nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002390(15a,17a-dimethyl-1-(1-propynyl)-(1R,15aS,17aS)-2,3...)
Affinity DataIC50:  180nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002461(10-Ethyl-1-[2-(3-ethyl-3H-benzothiazol-2-ylidene)-...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002389(1,15a,17a-trimethyl-(1S,15aS,17aS)-2,3,3a,3b,4,5,5...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002375(15a,17a-dimethyl-(1S,15aS,17aS)-2,3,3a,3b,4,5,5a,6...)
Affinity DataIC50:  220nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002460(1,3-Diethyl-2-[3-(3-ethyl-3H-benzooxazol-2-ylidene...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002464(10-Ethyl-1-[2-(1,1,3-trimethyl-1,3-dihydro-benzo[e...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002456(1,3-Diethyl-2-[3-(3-ethyl-3H-benzothiazol-2-yliden...)
Affinity DataIC50:  320nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002377(15a,17a-dimethyl-1-(2-propynyl)-(1R,15aS,17aS)-2,3...)
Affinity DataIC50:  320nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002378(1-(1-ethynyl)-17a,19a-dimethyl-(1R,5aS,17aS,19aS)-...)
Affinity DataIC50:  320nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009225(3-Ethyl-1-(3-hydroxy-propyl)-2-[3-(1,3,3-trimethyl...)
Affinity DataIC50:  350nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002459(1,3-Diethyl-2-[3-(1-ethyl-3,3-dimethyl-1,3-dihydro...)
Affinity DataIC50:  360nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009226(1,3-Diethyl-2-[3-(1-ethyl-3,3-dimethyl-1,3-dihydro...)
Affinity DataIC50:  390nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002458(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  390nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002457(1-(2-Acetoxy-ethyl)-3-ethyl-2-[3-(1,3,3-trimethyl-...)
Affinity DataIC50:  410nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009234(1-(3-Acetoxy-propyl)-3-ethyl-2-[3-(1,3,3-trimethyl...)
Affinity DataIC50:  410nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002452(3-Ethyl-1-(2-hydroxy-ethyl)-2-[3-(1,3,3-trimethyl-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002454(CHEMBL386306 | D-Lys(Nicotinoyl)-Pro(3-Pyridyl)-Al...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002454(CHEMBL386306 | D-Lys(Nicotinoyl)-Pro(3-Pyridyl)-Al...)
Affinity DataIC50:  500nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  510nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  510nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009235(1,3-Diethyl-2-[3-(3-methyl-3H-benzothiazol-2-ylide...)
Affinity DataIC50:  700nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002455(10-Ethyl-1-[2-(1,3,3-trimethyl-1,3-dihydro-indol-2...)
Affinity DataIC50:  790nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009227(1-(3-Ethoxycarbonyl-propyl)-3-ethyl-2-[3-(1,3,3-tr...)
Affinity DataIC50:  850nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009233(1,3-Diethyl-2-[3-(1-methyl-2a,5-dihydro-1H-benzo[c...)
Affinity DataIC50:  850nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009237(1,3-Diethyl-2-{3-[1-(2-hydroxy-ethyl)-3,3-dimethyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009231(6,7-Dichloro-1,3-diethyl-2-[3-(1,3,3-trimethyl-1,3...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002382(1-(1-ethynyl)-1-hydroxy-16a,18a-dimethyl-(1R,5aS,1...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002451(5-Ethyl-4-[2-(3-ethyl-3H-benzothiazol-2-ylidene)-e...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009236(1-(3-Dimethylamino-propyl)-3-ethyl-2-[3-(1,3,3-tri...)
Affinity DataIC50:  1.30E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009229(1-(3-Carboxy-propyl)-3-ethyl-2-[3-(1,3,3-trimethyl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002394(1-(1-ethynyl)-13a,15a-dimethyl-(1R,5aS,13aS,15aS)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009230(1,3-Diethyl-2-[3-(3-methyl-thiazolidin-2-ylidene)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity of compound was evaluated towards tachykinin receptor 2 by using radioligand ([125I]-NKA in rat duodenumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009232(1-Carbamoylmethyl-3-ethyl-2-[3-(1,3,3-trimethyl-1,...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002463(1,3-Diethyl-2-[3-(1-methyl-1H-benzo[cd]indol-2-yli...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002396(CHEMBL125109 | methyl 4-[4,17-dihydroxy-15a,17a-di...)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50009223(2-[3-(1-Dimethylcarbamoylmethyl-3,3-dimethyl-1,3-d...)
Affinity DataIC50:  2.60E+3nMAssay Description:Binding affinity for tachykinin receptor 1 from rat forebrain tissue, [125I]-BH-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002391(1-ethyl-15a,17a-dimethyl-(1S,15aS,17aS)-2,3,3a,3b,...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to standard Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  3.30E+3nMAssay Description:Binding affinity of compound was evaluated towards tachykinin receptor 3 by using radioligand [1261]eledoisin in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002453(10-Ethyl-1-[2-(3-ethyl-3H-benzooxazol-2-ylidene)-e...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002372(1,2,3,4-tetrahydrobenzo[4,5]imidazo[2,1-b]quinazol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002383(15a,17a-dimethyl-1-phenyl-(1S,15aS,17aS)-2,3,3a,3b...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002386(CHEMBL125493 | methyl 15a,17a-dimethyl-(1S,15aS,17...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125]I-Bolton Hunter Substance P([125]I-BHSP) binding to Tachykinin receptor 1 from rat forebrain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 64 total ) | Next | Last >>
Jump to: