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Found 30 with Last Name = 'lovas' and Initial = 's'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  0.00240nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  0.00950nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229425(CHEMBL401142 | Tyr-(R)-spiro-Aba-Gly-Phe-NH2)
Affinity DataKi:  0.0293nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229426(CHEMBL399796 | Tyr-(S)-Aba-Gly-Phe-NH2)
Affinity DataKi:  0.373nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataKi:  0.710nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229426(CHEMBL399796 | Tyr-(S)-Aba-Gly-Phe-NH2)
Affinity DataKi:  0.778nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229424(CHEMBL250448 | Tyr-(R)-Aba-Gly-Phe-NH2)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229427(CHEMBL401143 | Tyr-(S)-spiro-Aba-Gly-Phe-NH2)
Affinity DataKi:  2.31nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229424(CHEMBL250448 | Tyr-(R)-Aba-Gly-Phe-NH2)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229427(CHEMBL401143 | Tyr-(S)-spiro-Aba-Gly-Phe-NH2)
Affinity DataKi:  8.73nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229425(CHEMBL401142 | Tyr-(R)-spiro-Aba-Gly-Phe-NH2)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079406(Asp-Thr-D-Phe-Val-Gly-Leu-Nle-NH2 | Asp-Thr-Phe-Va...)
Affinity DataKi:  13nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataKi:  42nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079409(Asp-Thr-p-F-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL103634)
Affinity DataKi:  44nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  102nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079408(Asp-Thr-p-NH2-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL1039...)
Affinity DataKi:  156nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079410(Asp-Thr-p-Cl-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL10212...)
Affinity DataKi:  1.42E+3nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079407(Asp-Thr-Trp-Val-Gly-Leu-Nle-NH2 | CHEMBL319256)
Affinity DataKi: >2.00E+3nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50408715(CHEMBL2111616)
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity towards NK-2 receptors using [3H]NKA as radioligand in cloned human CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079411(Asp-Thr-p-NO2-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL4306...)
Affinity DataKi: >2.00E+3nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataIC50:  16.8nMAssay Description:Agonist activity at mu opioid receptor in NMRI mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079406(Asp-Thr-D-Phe-Val-Gly-Leu-Nle-NH2 | Asp-Thr-Phe-Va...)
Affinity DataIC50:  30.9nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50229425(CHEMBL401142 | Tyr-(R)-spiro-Aba-Gly-Phe-NH2)
Affinity DataIC50:  49.8nMAssay Description:Agonist activity at mu opioid receptor in NMRI mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Biological Research Center Of The Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataIC50:  75.5nMAssay Description:Agonist activity at mu opioid receptor in NMRI mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataIC50:  102nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079409(Asp-Thr-p-F-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL103634)
Affinity DataIC50:  107nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  245nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079408(Asp-Thr-p-NH2-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL1039...)
Affinity DataIC50:  372nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50079410(Asp-Thr-p-Cl-Phe-Val-Gly-Leu-Nle-NH2 | CHEMBL10212...)
Affinity DataIC50:  3.47E+3nMAssay Description:Inhibitory activity against human Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed