TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Cambridge
Curated by PDSP Ki Database
University Of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Cambridge
Curated by PDSP Ki Database
University Of Cambridge
Curated by PDSP Ki Database
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Cambridge
Curated by PDSP Ki Database
University Of Cambridge
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Cambridge
Curated by PDSP Ki Database
University Of Cambridge
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 0.823nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 1.02nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Cambridge
Curated by PDSP Ki Database
University Of Cambridge
Curated by PDSP Ki Database
Affinity DataKi: 1.40nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 1.52nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 2.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 2.32nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.38nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Cambridge
Curated by PDSP Ki Database
University Of Cambridge
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 2.92nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 3.61nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]diprenorphine from human MOR expressed in African green monkey COS1 cell membranes incubated for 1 hr by scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 7.74nMAssay Description:Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced responseMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 15.5nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 17.4nMAssay Description:Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced responseMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 27.2nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 29.6nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National University Of Singapore
Curated by ChEMBL
National University Of Singapore
Curated by ChEMBL
Affinity DataKi: 92.8nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair