TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 2.41nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Affinity of the compound for [3H]-N-propylnorapomorphine (NPA) Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 5.30nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibitory potency towards human cAPK C alpha in the presence of 100uM ATP and 30uM TAMRA-kemptideMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibitory potency towards human cAPK C alpha in the presence of 100uM ATP and 30uM TAMRA-kemptideMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 5.32nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibitory potency towards human cAPK C alpha in the presence of 100uM ATP and 30uM TAMRA-kemptideMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 8.30nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Institute Of Organic And Bioorganic Chemistry
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibitory potency towards human cAPK C alpha in the presence of 100uM ATP and 30uM TAMRA-kemptideMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Affinity of the compound for [3H]-N-propylnorapomorphine (NPA) Dopamine receptor D2More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 13.4nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 14.6nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Affinity for displacement of [3H]-WB-4101 labeled Dopamine receptor D1More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 21.1nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Concentration of the compound inhibiting specific binding of [3H]-haloperidol to Dopamine receptor D2 from rat striatal brain.More data for this Ligand-Target Pair
Affinity DataIC50: 30.7nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 36.9nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 43.1nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 54nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 56.6nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 97nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 100nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 123nMAssay Description:Concentration of the compound inhibiting specific binding of [3H]-haloperidol to Dopamine receptor D2 from rat striatal brain.More data for this Ligand-Target Pair
Affinity DataIC50: 409nMAssay Description:Affinity of the compound for [3H]-N-propylnorapomorphine (NPA) Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 409nMAssay Description:Concentration of the compound inhibiting specific binding of [3H]-haloperidol to Dopamine receptor D2 from rat striatal brain.More data for this Ligand-Target Pair
Affinity DataIC50: 662nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 774nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Concentration of the compound inhibiting specific binding of [3H]-haloperidol to Dopamine receptor D2 from rat striatal brain.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Affinity for displacement of [3H]-clonidine labeled Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: 1.61E+3nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 2.10E+3nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Mus musculus (mouse))
University Of Tartu
University Of Tartu
Affinity DataIC50: 2.60E+3nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 3.75E+3nMAssay Description:The IC50 values of the inhibitors corresponding to the concentration of the inhibitor decreasing the enzyme activity 50% were measured using fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for displacement of [3H]-clonidine labeled Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]-haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for displacement of [3H]-SCH-23,390 labeled Dopamine receptor D1More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Affinity for displacement of [3H]-WB-4101 labeled Dopamine receptor D1More data for this Ligand-Target Pair