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Found 2008 with Last Name = 'maerki' and Initial = 'hp'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140558(US8912221, 31)
Affinity DataKi:  0.600nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140539(US8912221, 12)
Affinity DataKi:  0.800nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140552(US8912221, 25)
Affinity DataKi:  1nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140550(US8912221, 23)
Affinity DataKi:  1nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140540(US8912221, 13)
Affinity DataKi:  1nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140567(US8912221, 40)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140542(US8912221, 15)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140571(US8912221, 44)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140532(US8912221, 5)
Affinity DataKi:  1.10nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140563(US8912221, 36)
Affinity DataKi:  1.20nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140551(US8912221, 24)
Affinity DataKi:  1.20nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140557(US8912221, 30)
Affinity DataKi:  1.30nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140570(US8912221, 43)
Affinity DataKi:  1.40nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140555(US8912221, 28)
Affinity DataKi:  1.40nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140541(US8912221, 14)
Affinity DataKi:  1.40nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140543(US8912221, 16)
Affinity DataKi:  1.60nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140547(US8912221, 20)
Affinity DataKi:  1.60nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140534(US8912221, 7)
Affinity DataKi:  1.60nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140549(US8912221, 22)
Affinity DataKi:  1.70nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140561(US8912221, 34)
Affinity DataKi:  2.20nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140559(US8912221, 32)
Affinity DataKi:  2.30nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140530(US8912221, 3)
Affinity DataKi:  2.40nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322986(CHEMBL1210141 | N-(1-((2,6-diethoxy-4'-(trifluorom...)
Affinity DataKi:  2.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322979(CHEMBL1210209 | N-(1-((2,6-diethoxy-4'-fluorobiphe...)
Affinity DataKi:  2.5nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140531(US8912221, 4)
Affinity DataKi:  2.5nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107177(US8592426, 26)
Affinity DataKi:  2.60nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140528(US8912221, 1)
Affinity DataKi:  2.60nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140538(US8912221, 11)
Affinity DataKi:  2.60nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140545(US8912221, 18)
Affinity DataKi:  3nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107189(US8592426, 38)
Affinity DataKi:  3nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50311334(2-(1-(4-chloro-3,5-diethoxybenzyl)piperidin-4-ylam...)
Affinity DataKi:  3nMAssay Description:Displacement of SST14 from human recombinant SST5 receptor expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107176(US8592426, 25)
Affinity DataKi:  3.10nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140562(US8912221, 35)
Affinity DataKi:  3.30nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107209(US8592426, 59)
Affinity DataKi:  3.5nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140564(US8912221, 37)
Affinity DataKi:  3.5nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107178(US8592426, 27)
Affinity DataKi:  3.60nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107203(US8592426, 53)
Affinity DataKi:  3.60nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107181(US8592426, 30)
Affinity DataKi:  3.90nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107193(US8592426, 42)
Affinity DataKi:  4nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322988(CHEMBL1210084 | N-(1-(3,5-diethoxy-4-methylbenzyl)...)
Affinity DataKi:  4nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107190(US8592426, 116 | US8592426, 117 | US8592426, 39/40...)
Affinity DataKi:  4nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107179(US8592426, 28)
Affinity DataKi:  4.10nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140565(US8912221, 38)
Affinity DataKi:  4.30nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140548(US8912221, 21)
Affinity DataKi:  4.30nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107163(US8592426, 12)
Affinity DataKi:  4.40nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107214(US8592426, 65)
Affinity DataKi:  4.40nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322981(CHEMBL1210207 | N-(1-((2,6-diethoxy-4'-fluorobiphe...)
Affinity DataKi:  4.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50322987(CHEMBL1210085 | N-(1-(4-chloro-3,5-diethoxybenzyl)...)
Affinity DataKi:  4.40nMAssay Description:Displacement of radio labeled 11 Tyr SST14 from human SST5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKininogen-1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM107206(US8592426, 56)
Affinity DataKi:  4.5nMAssay Description:Binding assay using Bradykinin-1 receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetB1 bradykinin receptor(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM140537(US8912221, 10)
Affinity DataKi:  4.70nMpH: 7.4Assay Description:For binding, Bradykinin-1 receptor antagonist compounds were added in various concentrations in 50 mM Tris pH 7.4, 5 mM MgCl2 together with 6 nM Kall...More data for this Ligand-Target Pair
In DepthDetails US Patent
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