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Found 84 with Last Name = 'malabre' and Initial = 'p'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368929(CHEMBL610155)
Affinity DataKi:  7nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453502(CHEMBL2113573)
Affinity DataKi:  7.5nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453499(CHEMBL2113598)
Affinity DataKi:  7.90nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368937(CHEMBL609252)
Affinity DataKi:  8.30nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453507(CHEMBL2113584)
Affinity DataKi:  11nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368950(CHEMBL610442)
Affinity DataKi:  14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368922(CHEMBL611311)
Affinity DataKi:  14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453512(CHEMBL2113599)
Affinity DataKi:  23nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211167(CHEMBL213255 | biphenyl-4-carboxylic acid [3-metho...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453510(CHEMBL2113586)
Affinity DataKi:  26nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453511(CHEMBL2113587)
Affinity DataKi:  29nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50150715(4''-Fluoro-biphenyl-4-carboxylic acid (6-dimethyla...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368940(CHEMBL611000)
Affinity DataKi:  39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368930(CHEMBL607875)
Affinity DataKi:  39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368931(CHEMBL608964)
Affinity DataKi:  50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368928(CHEMBL611600)
Affinity DataKi:  50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453500(CHEMBL2113596)
Affinity DataKi:  62nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211174(CHEMBL246588 | N-(3-methoxy-4-(2-(pyrrolidin-1-yl)...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211173(1-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  101nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453508(CHEMBL2113585)
Affinity DataKi:  110nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453501(CHEMBL2113597)
Affinity DataKi:  120nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368952(CHEMBL610717)
Affinity DataKi:  130nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368941(CHEMBL608369)
Affinity DataKi:  140nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368939(CHEMBL611598)
Affinity DataKi:  140nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453505(CHEMBL2113589)
Affinity DataKi:  150nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368943(CHEMBL609554)
Affinity DataKi:  160nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368951(CHEMBL611599)
Affinity DataKi:  160nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211166(1-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  164nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368953(CHEMBL608962)
Affinity DataKi:  170nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368947(CHEMBL610724)
Affinity DataKi:  170nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211160((Z)-5-(4-((3-hydroxypyrrolidin-1-yl)methyl)benzyli...)
Affinity DataKi:  176nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368927(CHEMBL609555)
Affinity DataKi:  180nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453504(CHEMBL2113591)
Affinity DataKi:  200nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211164((Z)-5-(4-(pyrrolidin-1-ylmethyl)benzylidene)-3-(4-...)
Affinity DataKi:  220nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211172(1-biphenyl-4-yl-3-[3-methoxy-4-(2-pyrrolidin-1-yl-...)
Affinity DataKi:  260nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211166(1-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  330nMAssay Description:Binding affinity to 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211176((Z)-5-(4-((dimethylamino)methyl)benzylidene)-3-(4-...)
Affinity DataKi:  341nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211168((Z)-5-(4-(azepan-1-ylmethyl)benzylidene)-3-(4-phen...)
Affinity DataKi:  357nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211170(3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  365nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453498(CHEMBL2113594)
Affinity DataKi:  370nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211166(1-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  370nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211161(3-biphenyl-4-yl-1-[3-methoxy-4-(2-pyrrolidin-1-yl-...)
Affinity DataKi:  415nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453509(CHEMBL2113603)
Affinity DataKi:  510nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211171((Z)-5-(4-((2-(dimethylamino)ethylamino)methyl)benz...)
Affinity DataKi:  707nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211166(1-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  880nMAssay Description:Binding affinity to 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453513(CHEMBL2113579)
Affinity DataKi:  890nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453503(CHEMBL2113590)
Affinity DataKi:  895nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211169(CHEMBL394311 | N-(3-methoxy-4-(2-(pyrrolidin-1-yl)...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Cerep

Curated by ChEMBL
LigandPNGBDBM50211163(1-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-...)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453506(CHEMBL2113583)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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