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Found 98 with Last Name = 'murai' and Initial = 'm'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM81444(CAS_185453 | NSC_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM31046(3-[4,5-dihydro-1H-imidazol-2-ylmethyl-(4-methylphe...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50033112(6-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyla...)
Affinity DataKi:  4.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM30712(6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimet...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM84342(4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...)
Affinity DataKi:  2.50E+3nMMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM84342(4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...)
Affinity DataKi:  4.80E+3nMMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM35234(DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradre...)
Affinity DataKi:  7.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50026777(2-Amino-1-(2,5-dimethoxy-phenyl)-propan-1-ol | 2-A...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92960(Piperazine derivative, 24)
Affinity DataIC50:  1nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92945(Piperazine derivative, 10)
Affinity DataIC50:  1.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411085(CHEMBL464549)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92946(Piperazine derivative, 9)
Affinity DataIC50:  1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92949(Piperazine derivative, 13)
Affinity DataIC50:  1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92955(Piperazine derivative, 19)
Affinity DataIC50:  2.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92948(Piperazine derivative, 12)
Affinity DataIC50:  2.30nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92941(Piperazine derivative, 5)
Affinity DataIC50:  2.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92950(Piperazine derivative, 14)
Affinity DataIC50:  2.80nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411084(CHEMBL208839)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92956(Piperazine derivative, 20)
Affinity DataIC50:  3.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92947(Piperazine derivative, 11)
Affinity DataIC50:  5.90nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411092(CHEMBL209302)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411088(CHEMBL211108)
Affinity DataIC50:  9nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92954(Piperazine derivative, 18)
Affinity DataIC50:  12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92944(Piperazine derivative, 8)
Affinity DataIC50:  12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50406796(CHEMBL2115161)
Affinity DataIC50:  13nMAssay Description:Tested for inhibition against [3H]-SP (substance P) (1 nM) binding to NK1 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033612(1H-Indole-2-carboxylic acid {5-(2-acetylamino-3-hy...)
Affinity DataIC50:  19nMAssay Description:Tested for inhibition against [3H]-SP (substance P) (1 nM) binding to NK1 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033610(1H-Indole-3-carboxylic acid {4-(2-acetylamino-3-hy...)
Affinity DataIC50:  21nMAssay Description:Tested for inhibition against [3H]-SP (substance P) (1 nM) binding to NK1 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033611(CHEMBL264384 | N*1*-[1-(Benzyl-methyl-carbamoyl)-2...)
Affinity DataIC50:  23nMAssay Description:Tested for inhibition against [3H]-SP (substance P) (1 nM) binding to NK1 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92942(Piperazine derivative, 6)
Affinity DataIC50:  26nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411091(CHEMBL377863)
Affinity DataIC50:  27nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411087(CHEMBL377013)
Affinity DataIC50:  34nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411082(CHEMBL208980)
Affinity DataIC50:  45nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411083(CHEMBL379529)
Affinity DataIC50:  45nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033609(CHEMBL306267 | N*1*-[1-(Benzyl-methyl-carbamoyl)-2...)
Affinity DataIC50:  54nMAssay Description:Tested for inhibition against [3H]-SP (substance P) (1 nM) binding to NK1 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002533(2-[2-(2-tert-Butoxycarbonylamino-4-carbamoyl-butyr...)
Affinity DataIC50:  90nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002552(CHEMBL303337 | benzyl 2-[2-(1-formyl-1H-3-indolyl)...)
Affinity DataIC50:  110nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002568(CHEMBL304472 | benzyl 2-[2-(1-formyl-1H-3-indolyl)...)
Affinity DataIC50:  110nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92943(Piperazine derivative, 7)
Affinity DataIC50:  110nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50033613(1H-Indole-2-carboxylic acid {4-(2-acetylamino-3-hy...)
Affinity DataIC50:  125nMAssay Description:Tested for inhibition against [3H]-SP (substance P) (1 nM) binding to NK1 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002543(CHEMBL59615 | benzyl 2-[2-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  140nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002562(CHEMBL294798 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  140nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002545(CHEMBL544284 | benzyl 2-[1-[1-amino-3-carbamoyl-(1...)
Affinity DataIC50:  210nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002571(CHEMBL293355 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  240nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002573(CHEMBL58245 | benzyl 2-[2-(1-formyl-1H-3-indolyl)-...)
Affinity DataIC50:  260nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411093(CHEMBL211884)
Affinity DataIC50:  280nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002563(CHEMBL62357 | benzyl 2-[1-[3-carbamoyl-1-neopentyl...)
Affinity DataIC50:  360nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002560(CHEMBL294814 | benzyl 2-[1-[3-carbamoyl-1-neopenty...)
Affinity DataIC50:  380nMAssay Description:Displacement of specific binding of [3H]SP to tachykinin receptor 1 from the isolated guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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