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Found 174 with Last Name = 'nakajima' and Initial = 'k'
TargetNeuromedin-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403793(CHEMBL2115415)
Affinity DataIC50:  0.720nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217526(CHEMBL366972)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50090485(CHEMBL295615 | spiro[(2-hydroxy)indane-1,40-piperi...)
Affinity DataIC50:  2.70nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217519(CHEMBL354709)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50057477(4-(3-{3-[(4-Isobutyl-benzyl)-(4-isobutyl-phenyl)-a...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibitory activity against human Steroid 5-alpha-reductase type 1 in COS-1 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403793(CHEMBL2115415)
Affinity DataIC50:  3.10nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217520(CHEMBL354645)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1 [89-488](Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM120757(US8703761, 1-29)
Affinity DataIC50:  3.5nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217517(CHEMBL353158)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469320(CHEMBL4293567)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469320(CHEMBL4293567)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His10-tagged ZZ-HCV3C-BRM ATPase-SnAC (636 to 1331 residues) (unknown origin) expressed in insect sf9 cells preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469324(CHEMBL4286345)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His10-tagged ZZ-HCV3C-BRM ATPase-SnAC (636 to 1331 residues) (unknown origin) expressed in insect sf9 cells preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469330(CHEMBL4295096)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469324(CHEMBL4286345)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469331(CHEMBL4282980)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His10-tagged ZZ-HCV3C-BRM ATPase-SnAC (636 to 1331 residues) (unknown origin) expressed in insect sf9 cells preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217511(CHEMBL172342)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469330(CHEMBL4295096)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His10-tagged ZZ-HCV3C-BRM ATPase-SnAC (636 to 1331 residues) (unknown origin) expressed in insect sf9 cells preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469329(CHEMBL4278436)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant His10-tagged ZZ-HCV3C-BRM ATPase-SnAC (636 to 1331 residues) (unknown origin) expressed in insect sf9 cells preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469331(CHEMBL4282980)
Affinity DataIC50: <5nMAssay Description:Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217506(CHEMBL170936)
Affinity DataIC50:  5.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217509(CHEMBL354731)
Affinity DataIC50:  5.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469329(CHEMBL4278436)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217508(CHEMBL367509)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217504(CHEMBL353284)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217505(CHEMBL414377)
Affinity DataIC50:  6.70nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217513(CHEMBL171658)
Affinity DataIC50:  6.80nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50090485(CHEMBL295615 | spiro[(2-hydroxy)indane-1,40-piperi...)
Affinity DataIC50:  6.80nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217528(CHEMBL353596)
Affinity DataIC50:  6.90nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50143817(CHEMBL3758618)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant 6His-tagged DAGT1 expressed in fall armyworm Sf9 cells using diolein and oleoyl-CoA incubated for 30 mins by LC/MS/MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217509(CHEMBL354731)
Affinity DataIC50:  7.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217505(CHEMBL414377)
Affinity DataIC50:  7.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217522(CHEMBL353394)
Affinity DataIC50:  7.80nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1 [89-488](Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM120755(US8703761, 1-8)
Affinity DataIC50:  8.5nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217507(CHEMBL171704)
Affinity DataIC50:  9.20nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217527(CHEMBL172227)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50239481(CHEMBL4061308)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217530(CHEMBL170084)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469325(CHEMBL4294655)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50469325(CHEMBL4294655)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant His10-tagged ZZ-HCV3C-BRM ATPase-SnAC (636 to 1331 residues) (unknown origin) expressed in insect sf9 cells preincubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1 [89-488](Homo sapiens (Human))
Novartis

US Patent
LigandPNGBDBM120756(US8703761, 1-28)
Affinity DataIC50:  11nMpH: 7.5 T: 2°CAssay Description:The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50143818(CHEMBL3759363)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant 6His-tagged DAGT1 expressed in fall armyworm Sf9 cells using diolein and oleoyl-CoA incubated for 30 mins by LC/MS/MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50057477(4-(3-{3-[(4-Isobutyl-benzyl)-(4-isobutyl-phenyl)-a...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory activity against human Steroid 5-alpha-reductase type 2 in COS-1 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403790(CHEMBL2114963)
Affinity DataIC50:  11nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]-SP from Tachykinin receptor 3 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217528(CHEMBL353596)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217519(CHEMBL354709)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217514(CHEMBL369246)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50239482(CHEMBL1683001)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217510(CHEMBL355387)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217512(CHEMBL169132)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50239480(CHEMBL4074410)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human His6-tagged DGAT1 expressed in Sf9 insect cell membranes assessed as inhibition of triglyceride formation using diole...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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