Affinity DataKi: 7.27E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+5nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.43E+6nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.47E+6nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.73E+6nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+7nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
TargetAcyl carrier protein,/NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial(Bos taurus)
Kyoto University
Curated by ChEMBL
Kyoto University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: >2.20E+4nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human intestinal sucrase in human Caco2 cell membraneMore data for this Ligand-Target Pair