Affinity DataKi: 0.0200nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 1 nM) calculated for the high affinity components of the [3H]spiroperidol b...More data for this Ligand-Target Pair
Affinity DataKi: 0.0310nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 1 uM) calculated for the high affinity components of the [3H]spiroperidol b...More data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of...More data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of...More data for this Ligand-Target Pair
Affinity DataKi: 0.0660nMAssay Description:Percentage of receptor in the low affinity form for the compound to Dopamine receptor D2 in absence of Gpp(NH)p (pre treated with 100 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 100 nM) calculated for the high affinity components of the [3H]spiroperidol...More data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0680nMAssay Description:Percentage of receptor in the high affinity form for the compound to Dopamine receptor D2 in presence of Gpp(NH)p (pretreated with 100 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.0710nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 100 nM) calculated for the high affinity components of the [3H]spiroperidol...More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of...More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.0980nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
Affinity DataKi: 0.122nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of...More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of...More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
Affinity DataKi: 0.196nMAssay Description:Inhibitor constant of compound for high affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of...More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Binding affinity against Opioid receptor mu 1 in Guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.980nMAssay Description:Binding affinity against Opioid receptor mu 1 in Guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.24nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Binding affinity against Opioid receptor kappa 1 in Guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for human placental microsome Cytochrome P450 19A1 by nonlinear regression analysisMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity for human placental microsome Cytochrome P450 19A1 by nonlinear regression analysisMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against Delta Opioid receptor in Guinea pig brain membranes using [3H]DAMGO+DADLEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Binding affinity against Kappa Opioid receptor in Guinea pig brain membranes using [3H]-DAMGO+EKCMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity for human placental microsome Cytochrome P450 19A1 by nonlinear regression analysisMore data for this Ligand-Target Pair
Affinity DataKi: 47.6nMAssay Description:Binding affinity for human placental microsome Cytochrome P450 19A1 by nonlinear regression analysisMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the low affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p (Pre treated with 1 nM) calculated for the high affinity components of the [3H]spiroperidol bi...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibitor constant of compound for low affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of ...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibitor constant of compound for low affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in presence of ...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the low affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p (Pre treated with 1 uM) calculated for the high affinity components of the [3H]spiroperidol bi...More data for this Ligand-Target Pair
Affinity DataKi: 60.1nMAssay Description:Inhibitor constant of compound for low affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of G...More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Percentage of receptor in the high affinity form for the compound to Dopamine receptor D2 in absence of Gpp(NH)p (pre treated with 1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 65.8nMAssay Description:Binding affinity for human placental microsome Cytochrome P450 19A1 by nonlinear regression analysisMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the low affinity components of the [3H]spiroperidol binding to Dopamine recepto...More data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the low affinity components of the [3H]spiroperidol binding to Dopamine recepto...More data for this Ligand-Target Pair
Affinity DataKi: 73.2nMAssay Description:Inhibitor constant of compound for low affinity component of [3H]-spiroperidol/N-propylnorapomorphine binding to Dopamine receptor D2 in absence of G...More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Percentage of receptor in the high affinity form for the compound to Dopamine receptor D2 in absence of Gpp(NH)p (pre treated with 1 uM)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Binding affinity against Kappa Opioid receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair