TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.00800nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0170nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 1 nM) calculated for the high affinity components of the [3H]spiroperidol b...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0220nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0250nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0260nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0270nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0360nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 1 uM) calculated for the high affinity components of the [3H]spiroperidol b...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0450nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0510nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.0660nMAssay Description:Percentage of receptor in the low affinity form for the compound to Dopamine receptor D2 in absence of Gpp(NH)p (pre treated with 100 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 100 nM) calculated for the high affinity components of the [3H]spiroperidol...More data for this Ligand-Target Pair
Affinity DataKi: 0.0680nMAssay Description:Percentage of receptor in the high affinity form for the compound to Dopamine receptor D2 in presence of Gpp(NH)p (pretreated with 100 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p (Pre treated with 100 nM) calculated for the high affinity components of the [3H]spiroperidol...More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.0980nMAssay Description:Inhibitory constant of compound in absence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recept...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.123nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.141nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.151nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibitory constant of compound in presence of Gpp(NH)p calculated for the high affinity components of the [3H]spiroperidol binding to Dopamine recep...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.229nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.257nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.309nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.525nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.525nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.661nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.708nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.832nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.840nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.871nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha7 using [3H]-MLA as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair