TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Inhibition of 1 nM [3H]- N6 -(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat fat cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.850nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.870nMAssay Description:Inhibition of [3H]- PIA binding at adenosine A1 receptor on rat cerebral cortex membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.900nMAssay Description:Inhibition of 1 nM [3H]- N6-(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of binding of [3H]nicotine to Nicotinic acetylcholine receptor alpha4-beta2 in rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:The compound was evaluated for percentage inhibition of binding of [3H]- nicotine to Nicotinic acetylcholine receptor alpha4-beta2 in Rat Cerebral Co...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Ability to inhibit the binding of [125I]physalaemin to the SP receptors in rat telencephalon slicesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Tested for the displacement [3H]-PIA from Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]- PIA binding at adenosine A1 receptor on rat cerebral cortex membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cerebral cortical membranes by [3H]-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Inhibition of 1 nM [3H]- N6 -(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat fat cell membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Inhibition of 1 nM [3H]- N6-(phenylisopropyl) adenosine binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibition of [3H]- oxotremorine-M binding to human Muscarinic acetylcholine receptor M4 in CHO cell membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cerebral cortical membranes by [3H]-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity against human recombinant Adenosine A3 receptor stably expressed in HEK293 cells by displacing [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Antagonism of binding of 1 nM [3H]cyclohexyladenosine to adenosine A1 receptors on rat cortical membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Binding affinity of the compound against A1 adenosine receptors of the central nervous systemMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Inhibition of binding of [3H]quinuclidinyl benzilate to muscarinic receptors in membranes of CHO cells transfected with Muscarinic acetylcholine rece...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Inhibition of [3H]- quinuclidinyl benzilate binding to human Muscarinic acetylcholine receptor M2 expressed in CHO cell membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Inhibition of binding of [3H]quinuclidinyl benzilate to Muscarinic acetylcholine receptor M2 in rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cerebral cortical membranes by [3H]-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Antagonism of binding of 1 nM [3H]cyclohexyladenosine to adenosine A1 receptors on rat cortical membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Binding affinity of the compound against A1 adenosine receptors of the central nervous systemMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 3.20nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]CP 55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 3.30nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]CP 55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]- oxotremorine-M binding to human Muscarinic acetylcholine receptor M4 in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]CP 55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cerebral cortical membranes by [3H]-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Ability to inhibit the binding of [3H]N6-phenylisopropyl adenosine to adenosine receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 4.5nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 4.5nMAssay Description:Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 4.60nMAssay Description:Binding affinity of the compound against A1 adenosine receptors of the central nervous systemMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Inhibition of [3H]- oxotremorine-M binding to human Muscarinic acetylcholine receptor M1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 5nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cerebral cortical membranes by [3H]-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute Of Diabetes
Curated by ChEMBL
National Institute Of Diabetes
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity against alpha 2-Adrenergic receptor in guinea pig cerebral cortical membranes by displacement of [3H]clonidineMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
National Institutes Of Diabetes And Digestive And Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]CP 55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair