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Found 162 with Last Name = 'perrakis' and Initial = 'a'
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50501623(CHEMBL4062929)
Affinity DataKi:  6nMAssay Description:Competitive inhibition of human ATX expressed in HEK293 Flp-In cells assessed as decrease in LPC hydrolysis measured every 30 secs for 90 mins by Lin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580260(CHEMBL5093347)
Affinity DataKi:  7nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Rattus norvegicus)
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50605406(CHEMBL5190935)
Affinity DataKi:  9nMAssay Description:Inhibition of rat ATX by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580262(CHEMBL5085520)
Affinity DataKi:  13nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580261(CHEMBL5084424)
Affinity DataKi:  14nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580256(CHEMBL5091502)
Affinity DataKi:  14nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580258(CHEMBL5076928)
Affinity DataKi:  15nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580255(CHEMBL5084058)
Affinity DataKi:  15nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580259(CHEMBL5088520)
Affinity DataKi:  15nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580263(CHEMBL5088371)
Affinity DataKi:  17nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580262(CHEMBL5085520)
Affinity DataKi:  19nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Rattus norvegicus)
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50605405(CHEMBL5196449)
Affinity DataKi:  24nMAssay Description:Inhibition of rat ATX by Michaelis-Menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM192943(US10526329, Compound 139 | US9670204, 138 2-((2-et...)
Affinity DataKi:  30nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580257(CHEMBL5078471)
Affinity DataKi:  32nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50580254(CHEMBL5088215)
Affinity DataKi:  41nMAssay Description:Inhibition of ATX lysoPLD (unknown origin) using 18:1 LPC as substrate assessed as reduction in choline release by HVA fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50267844(3-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-ylox...)
Affinity DataKi:  63.1nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  63.1nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50267883(8-Benzyl-3-(10,11-dihydro-5H-dibenzo[a,d]cyclohept...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413516(CHEMBL522249)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413513(CHEMBL452172)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413514(CHEMBL522981)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413509(CHEMBL523130)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413519(CHEMBL491860)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413520(CHEMBL503237)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413512(CHEMBL490643)
Affinity DataKi:  501nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413515(CHEMBL489034)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413517(CHEMBL490849)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR expressed in human SH-SY5Y cellsMore data for this Ligand-Target Pair
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413518(CHEMBL490442)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413510(HEPZIDINE)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50267844(3-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-ylox...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR expressed in human SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM50413511(CHEMBL489015)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
Institute

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acet...)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis His-tagged AchBPMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50267883(8-Benzyl-3-(10,11-dihydro-5H-dibenzo[a,d]cyclohept...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR expressed in human SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50233915(CHEMBL4102874)
Affinity DataIC50:  2nMAssay Description:Inhibition of ATX (unknown origin) using lysophosphatidyl choline as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50187693(CHEMBL3186509)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human ATX expressed in HEK293 cells using FS-3 as substrate preincubated for 15 mins followed by substrate addition measured after 30 m...More data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50187693(CHEMBL3186509)
Affinity DataIC50:  3nMAssay Description:Inhibition of human ATX expressed in HEK293 cells using FS-3 as substrate after 15 minsMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50187692(CHEMBL3827757)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human ATX using bisP-nitrophenyl phosphate as substrate measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50233913(CHEMBL4073215)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human ATX using bisP-nitrophenyl phosphate as substrate measured after 30 minsMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50347722(CHEMBL1802517)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50322727(4-[(4-{[3-(4-Fluorobenzyl)-2,4-dioxo-1,3-thiazolan...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50347723(CHEMBL1802518)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50347724(CHEMBL1802519)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50347716(CHEMBL1802471)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50347715(CHEMBL1802470)
Affinity DataIC50:  10nMAssay Description:Inhibition of 6x-histidine-tagged human recombinant ATX expressed in HEK293 cells assessed as choline release using lysophosphatidylcholine as substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50233919(CHEMBL4093897)
Affinity DataIC50:  11nMAssay Description:Inhibition of human ATX expressed in HEK293 Flp-In cells using LPC as substrate measured every 30 sec for 90 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Rattus norvegicus)
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50501623(CHEMBL4062929)
Affinity DataIC50:  20nMAssay Description:Inhibition of rat ATX lysoPLD activity using LPC as substrate assessed as reduction in choline release measured after 60 mins by HVA fluorescence bas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50501623(CHEMBL4062929)
Affinity DataIC50:  20nMAssay Description:Inhibition of human ATX expressed in HEK293 Flp-In cells assessed as decrease in choline release from LPC measured every 30 secs for 90 mins by HVA b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50187696(CHEMBL3621356)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant HA-tagged ATX (unknown origin) using FS-3 as substrate measured after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The Netherlands Institute

Curated by ChEMBL
LigandPNGBDBM50187692(CHEMBL3827757)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant human ATX using bisP-nitrophenyl phosphate as substrate measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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