Affinity DataKi: 0.0120nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta2 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0230nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta1 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 2.17E+5nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 4.93E+5nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
TargetThymidine kinase(Varicella-zoster virus (strain Dumas) (HHV-3) (Hum...)
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of VZV thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKd: 550nMAssay Description:Binding affinity to wild-type human partial length JAK1 JH2 pseudokinase domain (R537 to D855 residues) expressed in mammalian expression system at 1...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at rat adrenergic beta3 receptor expressed in DHB-11 CHO cells assessed as cAMP accumulation after 20 mins by scintillation proximit...More data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at human adrenergic beta3 receptor expressed in DHB-11 CHO cells assessed as cAMP accumulation after 20 mins by scintillation proxim...More data for this Ligand-Target Pair
TargetBone morphogenetic protein receptor type-1B(Homo sapiens (Human))
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataKd: 1.15E+4nMAssay Description:Binding affinity to BMPR1B by multi dose competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at human adrenergic beta1 receptor expressed in DHB-11 CHO cells assessed as cAMP accumulation after 20 mins by scintillation proxim...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataKd: 410nMAssay Description:Binding affinity to wild-type human partial length PIK3C3 (S282 to H879 residues) expressed in mammalian expression system at 10 uM by Kinomescan met...More data for this Ligand-Target Pair
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in DHB-11 CHO cells assessed as cAMP accumulation after 20 mins by scintillation proxim...More data for this Ligand-Target Pair