TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I]L-762,459 from recombinant human alpha1a adrenergic receptor expressed in mammalian cells measured after 1 hrMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]SNAP-7941 from recombinant human MCHR1 expressed in African green monkey COS7 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.43E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.68E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.11E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.22E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.42E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.49E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [3H]QNB from M1 receptor in Wistar rat cerebral cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.66E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.68E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.13E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.19E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.09E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.48E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.07E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.20E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.31E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.55E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.37E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 9.41E+4nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+5nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.29E+5nMAssay Description:Binding affinity to Toxoplasma gondii adenosine kinase after 20 mins by radioactivity methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Fyn (unknown origin) using Src-family kinase bisamide rhodamine 110 peptide substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Lyn (unknown origin) using Src-family kinase bisamide rhodamine 110 peptide substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Indo-Soviet Friendship College Of Pharmacy (Isfcp)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Src (unknown origin) using Src-family kinase bisamide rhodamine 110 peptide substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Antagonist activity at CCR4More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Antagonist activity at CCR4More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of GST-tagged PTP1B using pNPP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of MMP2 catalytic domain (unknown origin) using Ac-PLG-[2-mercapto-4-methylpentanoyl]-LG-OC2H5 as substrate preincubated for 45 to 120 min...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of COX2 (unknown origin) by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of COX2 (unknown origin) by EIAMore data for this Ligand-Target Pair
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of recombinant human LAT1More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis protein tyrosine phosphatase BMore data for this Ligand-Target Pair
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl alpha-d-glucopyranoside as substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human cytomegalovirus DNA polymerase (95 uL) activity in a solution containing 6.4 mM HEPES (pH 7.5), incubation for 12 minutes at 26 d...More data for this Ligand-Target Pair