TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg
Curated by ChEMBL
University Of Strasburg
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibition constant (Ki) against Human erythrocyte adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition constant (Ki) against Human erythrocyte adenosine deaminaseMore data for this Ligand-Target Pair
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg
Curated by ChEMBL
University Of Strasburg
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition constant (Ki) against calf intestine adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg
Curated by ChEMBL
University Of Strasburg
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition constant (Ki) against calf intestine adenosine deaminaseMore data for this Ligand-Target Pair
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg
Curated by ChEMBL
University Of Strasburg
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition constant (Ki) against Human erythrocyte adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition constant (Ki) against calf intestine adenosine deaminaseMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg
Curated by ChEMBL
University Of Strasburg
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg
Curated by ChEMBL
University Of Strasburg
Curated by ChEMBL
Affinity DataKi: 1.44E+3nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 4.63E+3nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 5.15E+3nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 8.23E+3nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.18E+4nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.35E+4nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition constant (Ki) against Human erythrocyte adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 2.12E+4nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+4nMAssay Description:Binding affinity against calf intestine adenosine deaminase enzymeMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 4.50E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 5.10E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
The University Of Tennessee Health Science Center
Curated by ChEMBL
The University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 5.76E+4nMAssay Description:Inhibition of N-terminal MKHQHQHQHQHQHQQPL-tagged 11beta-HSD1 C272S mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) using cortisol a...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 6.20E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 6.40E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.10E+4nMAssay Description:Inhibition constant (Ki) against calf intestine adenosine deaminaseMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 7.20E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 8.50E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 1.06E+5nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: 1.12E+5nMAssay Description:Displacement of [3H]dofetilide from human ERG by fliter binding assayMore data for this Ligand-Target Pair