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Found 103 with Last Name = 'rudo' and Initial = 'fg'
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.0200nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013943(CHEMBL327270 | Furan-2-carboxylic acid (2-chloro-p...)
Affinity DataKi:  0.130nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013945(CHEMBL431047 | Furan-2-carboxylic acid [3-methyl-1...)
Affinity DataKi:  0.150nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013934(CHEMBL319060 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  0.190nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013934(CHEMBL319060 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  0.190nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.220nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013939(CHEMBL95247 | Furan-2-carboxylic acid (3-methyl-1-...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013939(CHEMBL95247 | Furan-2-carboxylic acid (3-methyl-1-...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013938(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  0.330nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013938(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  0.330nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013949(CHEMBL95248 | Furan-2-carboxylic acid (2-methoxy-p...)
Affinity DataKi:  0.780nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013948(CHEMBL95909 | N-(2-Chloro-phenyl)-2-methoxy-N-(3-m...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  1.10nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017412(CHEMBL345120 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  1.90nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013935(CHEMBL95390 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-m...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013947(CHEMBL95786 | Furan-2-carboxylic acid (2-methoxy-p...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013940(CHEMBL319343 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-...)
Affinity DataKi:  2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  2.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  2.20nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017406(CHEMBL162700 | Furan-3-carboxylic acid benzo[1,2,5...)
Affinity DataKi:  2.60nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013942(CHEMBL318895 | N-(2-Chloro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  2.80nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228269(CHEMBL178035)
Affinity DataKi:  3.5nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017416(CHEMBL347188 | Furan-2-carboxylic acid (4-methyl-p...)
Affinity DataKi:  4.10nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013936(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013936(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017404(CHEMBL161084 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  7.5nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013944(2-Methoxy-N-(2-methoxy-phenyl)-N-(3-methyl-1-phene...)
Affinity DataKi:  7.60nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017420(CHEMBL157922 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  7.70nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228255(CHEMBL362439)
Affinity DataKi:  7.70nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013941(CHEMBL99596 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-m...)
Affinity DataKi:  8.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM83450(ALFENTANIL | Alfentanil hydrochloride | MLS0023206...)
Affinity DataKi:  8.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228260(CHEMBL367286)
Affinity DataKi:  8.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM83450(ALFENTANIL | Alfentanil hydrochloride | MLS0023206...)
Affinity DataKi:  8.20nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017403(CHEMBL161442 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  8.40nMAssay Description:The ability of the compound to displace [3H]-naloxone from the opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228221(CHEMBL366899)
Affinity DataKi:  9.10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228224(CHEMBL367667)
Affinity DataKi:  10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228217(CHEMBL174694)
Affinity DataKi:  10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013937(2-Methoxy-N-(2-methoxy-phenyl)-N-[3-methyl-1-(2-th...)
Affinity DataKi:  11nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228259(CHEMBL426034)
Affinity DataKi:  12nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017405(2-Methoxy-N-(1-phenethyl-piperidin-4-yl)-N-pyridin...)
Affinity DataKi:  13nMAssay Description:The ability of the compound to displace [3H]-naloxone from the Opioid receptor mu isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228251(CHEMBL176438)
Affinity DataKi:  14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228219(CHEMBL178847)
Affinity DataKi:  14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017411(CHEMBL158857 | Furan-2-carboxylic acid (1-phenethy...)
Affinity DataKi:  14nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017410(2-Methoxy-N-(1-phenethyl-piperidin-4-yl)-N-pyrimid...)
Affinity DataKi:  16nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017409(CHEMBL161023 | Furan-2-carboxylic acid (6-chloro-p...)
Affinity DataKi:  19nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017414(CHEMBL161147 | Furan-3-carboxylic acid (2-chloro-p...)
Affinity DataKi:  21nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50017413(CHEMBL161082 | Furan-2-carboxylic acid (2-chloro-p...)
Affinity DataKi:  22nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228218(CHEMBL368487)
Affinity DataKi:  24nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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