TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0190nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.172nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.208nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.248nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.75nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 9.37nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 13.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 20.0nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 24.9nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 36.6nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 41.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 54.2nMAssay Description:Displacement of [125I]IMSB from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 55.9nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 233nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 316nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 839nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Sungkyunkwan University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 958nMAssay Description:Displacement of [125I]IMPY from beta amyloid protein 40More data for this Ligand-Target Pair
Affinity DataIC50: 50.6nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.92E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 5.18E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig assessed as inhibition of electrically evoked-contractionMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 1.64E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 3.22E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 5.27E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Korea Basic Science Institute (Kbsi)
Curated by ChEMBL
Affinity DataIC50: 7.10E+4nMAssay Description:Displacement of 5-carboxyfluorescein-labeled PBD-binding peptide from PLk1 PBD (unknown origin) expressed in bacterial expression system incubated fo...More data for this Ligand-Target Pair