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Found 19 with Last Name = 'salo-ahen' and Initial = 'om'
TargetThymidylate synthase(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of thymidin synthaseMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of DHFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM50326711(1,3-propanediphosphonic acid | CHEMBL1230579 | PRO...)
Affinity DataKi:  260nMAssay Description:Inhibition of human Thymidylate synthase by uncompetitive bindingMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM18796((2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-...)
Affinity DataKi:  380nMAssay Description:Inhibition of GARFTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM50326711(1,3-propanediphosphonic acid | CHEMBL1230579 | PRO...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of human Thymidylate synthase by noncompetitive bindingMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM50326712(2(R)-[4(S)-carboxy-4-[4-[N-(2-hydroxymethyl-4-oxo-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of ERalpha expressed in human tumor cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Institute Of Theoretical Studies Ggmbh

Curated by ChEMBL
LigandPNGBDBM50326712(2(R)-[4(S)-carboxy-4-[4-[N-(2-hydroxymethyl-4-oxo-...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of thymidin synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM26739(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191457(4-(thiazol-2-yl)phenyl butylcarbamate | CHEMBL3767...)
Affinity DataIC50:  520nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191456(1-(2-phenyl-1,3-thiazol-4-yl)ethanone [4-(4-methyl...)
Affinity DataIC50:  690nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191459(4-[4-(benzyloxy)phenyl]-5-[(5-nitro-1,3-thiazol-2-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191462(1-(3-methyl-1-benzothien-2-yl)ethanone O-(anilinoc...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191461(1-(4-fluorophenyl)-2-(1-(4-hydroxyphenyl)-1H-tetra...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191454(1-(4-((4-(2,5-dimethyl-1-(thiophen-2-ylmethyl)-1H-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191455(CHEMBL213901 | ethyl 2-(2-(3-(styrylthio)propanami...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191457(4-(thiazol-2-yl)phenyl butylcarbamate | CHEMBL3767...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of MGL-like activity in Wistar rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191458(4-[4-(benzyloxy)phenyl]-3-methyl-5-[(5-nitro-1,3-t...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50191460((2-((6-methylpyridin-3-yloxy)methyl)morpholino)(2-...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of Wistar rat brain FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed