TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Research Center Idrtech
Curated by ChEMBL
Research Center Idrtech
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Inje University
Curated by ChEMBL
Inje University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Dyrk1 (unknown origin) autophosphorylationMore data for this Ligand-Target Pair