Compile Data Set for Download or QSAR
maximum 50k data
Found 943 with Last Name = 'stalder' and Initial = 'h'
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109401(US8604061, 115)
Affinity DataKi:  0.100nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109462(US8604061, 201)
Affinity DataKi:  0.200nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109373(US8604061, 48)
Affinity DataKi:  0.200nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109408(US8604061, 127)
Affinity DataKi:  0.300nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109581(US8604061, 316)
Affinity DataKi:  0.300nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109564(US8604061, 354)
Affinity DataKi:  0.300nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109528(US8604061, 298)
Affinity DataKi:  0.400nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109390(US8604061, 103)
Affinity DataKi:  0.400nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109580(US8604061, 296)
Affinity DataKi:  0.400nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109446(US8604061, 178)
Affinity DataKi:  0.400nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109356(US8604061, 14)
Affinity DataKi:  0.5nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109441(US8604061, 168)
Affinity DataKi:  0.600nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109576(US8604061, 374)
Affinity DataKi:  0.600nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109388(US8604061, 91)
Affinity DataKi:  0.600nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109504(US8604061, 256)
Affinity DataKi:  0.600nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109488(US8604061, 232)
Affinity DataKi:  0.600nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109420(US8604061, 143)
Affinity DataKi:  0.700nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109392(US8604061, 105)
Affinity DataKi:  0.700nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109411(US8604061, 132)
Affinity DataKi:  0.700nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109367(US8604061, 33)
Affinity DataKi:  0.700nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109384(US8604061, 86)
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109523(US8604061, 291)
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109379(US8604061, 80 (S))
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109362(US8604061, 21 (S))
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109548(US8604061, 330)
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109454(US8604061, 190)
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109453(US8604061, 189)
Affinity DataKi:  0.800nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109535(US8604061, 308)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109573(US8604061, 369)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109426(US8604061, 150)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109413(US8604061, 135)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106590(US8586617, 51)
Affinity DataKi:  0.900nM ΔG°:  -48.0kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109509(US8604061, 265)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109476(US8604061, 219)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109361(US8604061, 20)
Affinity DataKi:  0.900nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109434(US8604061, 159)
Affinity DataKi:  1nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106641(US8586617, 225)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109386(US8604061, 88)
Affinity DataKi:  1nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109572(US8604061, 367)
Affinity DataKi:  1nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109490(US8604061, 235)
Affinity DataKi:  1nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM47082(CHEMBL2206377 | US8586617, 24)
Affinity DataKi:  1nMAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106672(US8586617, 333)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106671(US8586617, 331)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106667(US8586617, 312)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106665(US8586617, 308)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106661(CHEMBL2206385 | US8586617, 304)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106660(US8586617, 303)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106658(US8586617, 297)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM106655(US8586617, 291)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/moleT: 2°CAssay Description:Radioligand binding assay: The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-1-naphthyl)-2-imidazoline was used at a concentration equal to the calcula...More data for this Ligand-Target Pair
In DepthDetails US Patent
Displayed 1 to 50 (of 943 total ) | Next | Last >>
Jump to: