Affinity DataKi: 0.0180nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0230nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0240nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0330nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0870nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal dopamine receptor D2 was determined in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal dopamine receptor D2 was determined in vitroMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 17.9nMAssay Description:Displacement of [3H]AZD9272 from human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counterMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]MPEP from human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Klinikum Der Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair