Affinity DataKi: 0.640nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 in rat adrenal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity was evaluated towards Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:The ability to displace [3H]clonidine from the Alpha-2 adrenergic receptor was determined in rat brain membraneMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-rosiglitazone from GST-tagged PPARgammaLBD (unknown origin) after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Ki value was evaluated against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Ki value was evaluated against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Ki value was evaluated against Angiotensin II receptor, type 2More data for this Ligand-Target Pair
Affinity DataKi: 730nMAssay Description:Ki value was evaluated against Angiotensin II receptor, type 2More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.58E+4nMAssay Description:The ability to displace [3H]clonidine from the Alpha-2 adrenergic receptor was determined in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity was evaluated against Angiotensin II receptor, type 1 in rabbit aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity for Angiotensin II receptor, type 1More data for this Ligand-Target Pair