Compile Data Set for Download or QSAR
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Found 451 with Last Name = 'tolman' and Initial = 'rl'
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002151(8-Piperazin-1-yl-imidazo[1,2-a]pyrazine | CHEMBL33...)
Affinity DataKi:  15nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002156(2-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  51nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002155(6-Chloro-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  73nMAssay Description:Binding affinity against alpha-2 adrenergic receptor was determined in calf cerebral cortex homogenates using [3H]clonidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002145(5-Methyl-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a...)
Affinity DataKi:  81nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002142(5-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  140nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002146(3,6-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  150nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002150(5-Bromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazine | ...)
Affinity DataKi:  170nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002150(5-Bromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazine | ...)
Affinity DataKi:  182nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002152(6-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  190nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002152(6-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  220nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002144(3-Chloro-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  240nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002139(3-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  240nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002155(6-Chloro-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  250nMAssay Description:Inhibition of human carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002146(3,6-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  250nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002154(5-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)
Affinity DataKi:  270nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002152(6-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  280nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002156(2-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  310nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002138(3,5-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  340nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002142(5-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  360nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002149(3-Isopropyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  370nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002151(8-Piperazin-1-yl-imidazo[1,2-a]pyrazine | CHEMBL33...)
Affinity DataKi:  400nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002138(3,5-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  400nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002147(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  480nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002154(5-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)
Affinity DataKi:  500nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002150(5-Bromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazine | ...)
Affinity DataKi:  520nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002143(3-Ethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; 2...)
Affinity DataKi:  530nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002146(3,6-Dimethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazi...)
Affinity DataKi:  620nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002157(3,5-Dibromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  630nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002142(5-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  820nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002148(8-Piperazin-1-yl-2,3-dihydro-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  870nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002153(8-(4-Methyl-piperazin-1-yl)-imidazo[1,2-a]pyrazine...)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002140(3-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)
Affinity DataKi:  1.35E+3nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002147(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  1.39E+3nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002141(3-Methyl-8-piperazin-1-yl-2,3-dihydro-imidazo[1,2-...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002151(8-Piperazin-1-yl-imidazo[1,2-a]pyrazine | CHEMBL33...)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002149(3-Isopropyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  2.01E+3nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002139(3-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002139(3-Methyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002145(5-Methyl-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002149(3-Isopropyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  2.99E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002143(3-Ethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; 2...)
Affinity DataKi:  3.24E+3nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002143(3-Ethyl-8-piperazin-1-yl-imidazo[1,2-a]pyrazine; 2...)
Affinity DataKi:  5.00E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002140(3-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002147(8-Piperazin-1-yl-3-propyl-imidazo[1,2-a]pyrazine; ...)
Affinity DataKi:  7.79E+3nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002141(3-Methyl-8-piperazin-1-yl-2,3-dihydro-imidazo[1,2-...)
Affinity DataKi:  1.03E+4nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002157(3,5-Dibromo-8-piperazin-1-yl-imidazo[1,2-a]pyrazin...)
Affinity DataKi:  1.19E+4nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002141(3-Methyl-8-piperazin-1-yl-2,3-dihydro-imidazo[1,2-...)
Affinity DataKi:  1.77E+4nMAssay Description:Binding affinity against Beta-2 adrenergic receptor was measured using [125I]CYP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032773((4aR,6aS)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032782((4aR,6aS)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032789((4aR,6aS)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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