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Found 41 with Last Name = 'tottori' and Initial = 'k'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  9.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  18.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM82065(CAS_163839 | NSC_163839 | OPC-4392)
Affinity DataKi:  19.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Third Tokushima Institute Of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  46.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084312((+)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(2-prope...)
Affinity DataIC50:  50nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes (high)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084320(5-Chloro-1-{3-[4-(3-methoxy-phenyl)-piperazin-1-yl...)
Affinity DataIC50:  130nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084310(1-{3-[4-(3-Bromo-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  150nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50369619(CHEMBL1743967)
Affinity DataIC50:  240nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084307(1-{3-[4-(2-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  260nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084325(5-Chloro-1-{3-[4-(3-propoxy-phenyl)-piperazin-1-yl...)
Affinity DataIC50:  370nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084313(5-Chloro-1-{3-[4-(3-nitro-phenyl)-piperazin-1-yl]-...)
Affinity DataIC50:  390nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM81982(CAS_97-39-2 | DITOLYLGUANIDINE | DTG | Di-o-tolylg...)
Affinity DataIC50:  400nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084308(1-{3-[4-(3-Bromo-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  420nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084324(1-{3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  460nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084311(5-Methoxy-1-{3-[4-(3-trifluoromethyl-phenyl)-piper...)
Affinity DataIC50:  490nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084321(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  600nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084326(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  620nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084329(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  650nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084323(CHEMBL299492 | N-(3-{4-[3-(5-Chloro-2-oxo-3,4-dihy...)
Affinity DataIC50:  670nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084319(1-{3-[4-(3-Amino-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  710nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084315(1-{3-[4-(3-Hydroxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataIC50:  810nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084305(5-Methoxy-1-{3-[4-(3-trifluoromethyl-phenyl)-piper...)
Affinity DataIC50:  820nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084316(1-(4-Fluoro-phenyl)-4-(5-fluoro-pyridin-2-yl)-4-pi...)
Affinity DataIC50:  860nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084322(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  870nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084306(5-Methoxy-1-{3-[4-(3-nitro-phenyl)-piperazin-1-yl]...)
Affinity DataIC50:  870nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084309(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  980nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084330(1-{3-[4-(3-Chloro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  1.13E+3nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084327(1-{3-[4-(3-Amino-phenyl)-piperazin-1-yl]-propyl}-5...)
Affinity DataIC50:  1.21E+3nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084317(1-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataIC50:  1.32E+3nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084331(3-{4-[3-(5-Methoxy-2-oxo-3,4-dihydro-2H-quinolin-1...)
Affinity DataIC50:  2.47E+3nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50019742(9-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)-9...)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084312((+)-1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(2-prope...)
Affinity DataIC50:  8.94E+3nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes (low)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084328(Benzoic acid 2-oxo-1-[3-(4-phenyl-piperazin-1-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084314(CHEMBL56373 | N-(7-Hydroxy-2,2,4,6-tetramethyl-ind...)
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity for sigma receptor was evaluated by the inhibitory effect on [3H]DTG to rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed