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Found 488 with Last Name = 'vacondio' and Initial = 'f'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.166nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541723(CHEMBL4649122)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50156100(CHEMBL3780550)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.295nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50156101(CHEMBL3780075)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419598(CHEMBL1934049)
Affinity DataKi:  0.372nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419584(CHEMBL1934062)
Affinity DataKi:  0.513nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50156023(CHEMBL3780521)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419598(CHEMBL1934049)
Affinity DataKi:  0.661nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50272462(CHEMBL525528 | N-(Adamant-1-yl)-7-fluoro-4-oxo-1-p...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419595(CHEMBL1934061)
Affinity DataKi:  0.871nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541729(CHEMBL4637535)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50156024(CHEMBL3780852)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50156022(CHEMBL3780166)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419588(CHEMBL1934057)
Affinity DataKi:  1.26nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419582(CHEMBL1934064)
Affinity DataKi:  1.26nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419597(CHEMBL1934053)
Affinity DataKi:  1.29nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541727(CHEMBL4647226)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419588(CHEMBL1934057)
Affinity DataKi:  1.41nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419585(CHEMBL1934060)
Affinity DataKi:  1.48nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419593(CHEMBL1934048)
Affinity DataKi:  1.48nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419596(CHEMBL1934056)
Affinity DataKi:  1.55nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50272486(CHEMBL498527 | N-(Adamant-1-yl)-4-oxo-1-pentyl-7-(...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50066960(CHEMBL33700 | N-(2-(5-methoxy-1-methyl-1H-indol-3-...)
Affinity DataKi:  1.70nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419595(CHEMBL1934061)
Affinity DataKi:  1.78nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50200170(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541725(CHEMBL4635230)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419585(CHEMBL1934060)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419581(CHEMBL1934065)
Affinity DataKi:  2.04nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419581(CHEMBL1934065)
Affinity DataKi:  2.09nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541721(CHEMBL4633927)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50066960(CHEMBL33700 | N-(2-(5-methoxy-1-methyl-1H-indol-3-...)
Affinity DataKi:  2.20nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419579(CHEMBL1934054)
Affinity DataKi:  2.34nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419586(CHEMBL1934059)
Affinity DataKi:  2.45nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419589(CHEMBL1934055)
Affinity DataKi:  2.45nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541737(CHEMBL4640659)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419583(CHEMBL1934063)
Affinity DataKi:  2.57nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419587(CHEMBL1934058)
Affinity DataKi:  3.02nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419593(CHEMBL1934048)
Affinity DataKi:  3.55nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50272510(CHEMBL523577 | N-(Adamant-1-yl)-4-oxo-1-pentyl-6-p...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419597(CHEMBL1934053)
Affinity DataKi:  4.27nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419583(CHEMBL1934063)
Affinity DataKi:  4.68nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50180040(4-Oxo-1-pentyl-1,4-dihydro-quinoline-3-carboxylic ...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541732(CHEMBL4636524)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50272486(CHEMBL498527 | N-(Adamant-1-yl)-4-oxo-1-pentyl-7-(...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50200170(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419590(CHEMBL1934052)
Affinity DataKi:  5.62nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50541722(CHEMBL4641997)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50272388(6-Isopropyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-CP-55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by Competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50471835(CHEMBL34327)
Affinity DataKi:  6.5nMAssay Description:Binding Affinity (pKi) towards human Melatonin receptor type 1BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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