Affinity DataKi: 2.40nM Kon: 0.000300M-1s-1 Koff: 1.40E+5s-1Assay Description:Compound was evaluated for the enzyme kinetic data (kon) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
Affinity DataKi: 3nM Kon: 0.00200M-1s-1 Koff: 7.00E+5s-1Assay Description:Compound was evaluated for the enzyme kinetic data (kon) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
Affinity DataKi: 3nM Kon: 0.000700M-1s-1 Koff: 2.30E+5s-1Assay Description:Compound was evaluated for the enzyme kinetic data (kon) for binding inhibition against Prolyl Endopeptidase (PEP)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for binding inhibition against Prolyl Endopeptidase (PEP).More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Inhibition of [3H]- rolipram binding to phosphodiesterase 4 of rat cerebral cortex membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Inhibition of [3H]- rolipram binding to rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE).More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE)More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE).More data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for displacement of radiolabelled [I-125]GRP from rat brain receptor; 1.5-3 microMMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for displacement of radiolabelled [I-125]GRP from rat brain receptor; 1.5-3 microMMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of calcium-independent Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]NT from the neurotensin receptor of bovine brainMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of cAMP-specific calcium-independent phosphodiesterase (IPDE)More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration required for the displacement of [3H]-NT from neurotensin receptor in mouse; value ranges from 4-6 microMMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of [3H]rolipram binding to rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of [3H]cAMP (NEN NET-275) binding to Calcium-Independent Phosphodiesterase from rat brain.More data for this Ligand-Target Pair