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Found 729 with Last Name = 'virone-oddos' and Initial = 'a'
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039364(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039345(CHEMBL77783 | Methyl-{5-methyl-7-propyl-8-[2'-(1H-...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039376(CHEMBL80773 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039366(2-(2-Hydroxy-ethyl)-5-methyl-7-propyl-8-[2'-(1H-te...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368929(CHEMBL610155)
Affinity DataKi:  7nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453502(CHEMBL2113573)
Affinity DataKi:  7.5nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453499(CHEMBL2113598)
Affinity DataKi:  7.90nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039344(2-Ethyl-5-methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368937(CHEMBL609252)
Affinity DataKi:  8.30nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039372(CHEMBL80380 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039362(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039341(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039350(5-Hydroxymethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039378(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453507(CHEMBL2113584)
Affinity DataKi:  11nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039346(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039374(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039357(CHEMBL312632 | {5-Methyl-3-oxo-7-propyl-8-[2'-(1H-...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368922(CHEMBL611311)
Affinity DataKi:  14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368950(CHEMBL610442)
Affinity DataKi:  14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039347(2-Methoxymethyl-5-methyl-7-propyl-8-[2'-(1H-tetraz...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453512(CHEMBL2113599)
Affinity DataKi:  23nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039368(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039342(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453510(CHEMBL2113586)
Affinity DataKi:  26nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039371(CHEMBL76149 | {2-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039370(2-Methoxy-5-methyl-7-propyl-8-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453511(CHEMBL2113587)
Affinity DataKi:  29nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039351(7-Butyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039352(CHEMBL80967 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039369(2,5-Dimethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039365(7-Ethyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039339(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368940(CHEMBL611000)
Affinity DataKi:  39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368930(CHEMBL607875)
Affinity DataKi:  39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039348(2-[4-(5-Methyl-3-oxo-7-propyl-2,3-dihydro-[1,2,4]t...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039375(7-Propyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  46nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368931(CHEMBL608964)
Affinity DataKi:  50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039354(7-Propyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368928(CHEMBL611600)
Affinity DataKi:  50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039361(2,5-Dimethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453500(CHEMBL2113596)
Affinity DataKi:  62nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039358(7-Cyclopropyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-bi...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039379(5-Methoxymethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataKi:  92nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039363(CHEMBL80161 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  99nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039373(7-Butyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  106nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453508(CHEMBL2113585)
Affinity DataKi:  110nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039343(5-Methoxymethyl-2-methyl-7-propyl-8-[2'-(1H-tetraz...)
Affinity DataKi:  111nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453501(CHEMBL2113597)
Affinity DataKi:  120nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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