Affinity DataKi: 0.700nMAssay Description:Binding affinity to Sigma opioid receptor type 1 in guinea pig brain homogenate with 0.5 nM of [3H](+)-PENT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity to Sigma opioid receptor type 2 in guinea pig brain homogenate with 4 nM of [3H](+)-DTG as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
Affinity DataKi: 220nMAssay Description:Compound was evaluated for its inhibitory constant against 3-dehydroquinate synthaseMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
Affinity DataKi: 250nMAssay Description:Compound was tested for inhibitory activity against FK506 binding protein 12 (FKBP12)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Pfizer
Curated by PDSP Ki Database
Pfizer
Curated by PDSP Ki Database