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Found 646 with Last Name = 'west' and Initial = 're'
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50264895(5-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)phenyl)-2...)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells assessed as reversal of N-alpha-methylhistamine-induced inhibition of fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325449(1-(2-(piperidin-1-yl)ethyl)-3-(1-(1-(pyridin-4-ylm...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175828(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325450(1-(2-(dimethylamino)ethyl)-3-(1-(1-(pyridin-4-ylme...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325466(1-(3-(dimethylamino)propyl)-3-(1-(1-(pyridin-4-ylm...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325465(1-benzyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-4-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175843(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325460(1-(4-methoxybenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pi...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325461(1-(3-methoxybenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pi...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175833(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175843(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325473(1-isobutyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | N-alpha-methylhistamine...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325448(1-(2-morpholinoethyl)-3-(1-(1-(pyridin-4-ylmethyl)...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441652(CHEMBL2437433)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441649(CHEMBL2437416)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325469(1-(2-isopropoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441646(CHEMBL2437421)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325467(1-(3-ethoxypropyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325462(1-(4-chlorobenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441637(CHEMBL2437430)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325472(1-(2-hydroxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177543(1-(3-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50264934(5-fluoro-2-(pyridin-2-yl)-1-(4-(3-(pyrrolidin-1-yl...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM22904((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50264895(5-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)phenyl)-2...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441642(CHEMBL2437425)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441647(CHEMBL2437420)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175833(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325470(1-(2-ethoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pipe...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50265014(1-(3-(4-(5-fluoro-2-(pyridin-2-yl)-1H-benzo[d]imid...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50264895(5-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)phenyl)-2...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to mouse histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86188(CHEMBL366977 | SCH 79687)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175828(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325451(1-(1-(1-(pyridin-4-ylmethyl)piperidine-4-carbonyl)...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175846(4-((1H-imidazol-4-yl)methyl)-1-(3-(3-chlorophenoxy...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175836(CHEMBL200643 | N-(3-(4-((1H-imidazol-4-yl)methyl)p...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175827(4-((1H-imidazol-4-yl)methyl)-1-heptylpiperidine | ...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50264932(1-(4-(3-(4-benzylpiperidin-1-yl)propoxy)phenyl)-5-...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in HEK cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325463(1-(3-chlorobenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50314290(3-benzyl-1-(4-bromophenyl)-1-(1-(pyridin-4-ylmethy...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human recombinant histamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175851(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-p...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325471(1-(2-methoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325468(1-(2-phenoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50383459(CHEMBL2031619)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human histamine H3 receptor expressed in HEK cell membranes after 30 mins by scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441641(CHEMBL2437426)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441645(CHEMBL2437422)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50383442(CHEMBL2031602)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50441654(CHEMBL2437431)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-N-alpha-methyl histamine from histamine H3 receptor in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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