Affinity DataKi: 0.0130nMAssay Description:Inhibitory activity of the compound against Coagulation factor Xa (serine protease) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Tested for binding affinity against human Coagulation factor Xa (trypsin-like serine protease)More data for this Ligand-Target Pair
Affinity DataKi: 0.0440nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 0.105nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibitory activity of the compound against factor Xa,activity expressed as Ki nMMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:In vitro inhibitory activity against serine protease thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro inhibitory activity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Binding affinity of the compound towards factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro inhibitory activity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro inhibitory activity of the compound against Coagulation factor X was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:In vitro inhibitory activity against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Tested for inhibitory activity against Coagulation factor Xa (trypsin-like serine protease) of the compoundMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Tested for the binding affinity against trypsinMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Tested for the binding affinity against thrombinMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:In vitro inhibitory activity against coagulation factor XMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against factor XaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Factor 10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against factor XaMore data for this Ligand-Target Pair