Affinity DataKi: 0.300nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]mibolerone from Androgen receptor (unknown origin) measured by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity to human BRD2 BD1 (72 to 205 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Agonist activity at Androgen receptor expressed in mouse C2C12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity to human BRD3 BD1 (24 to 144 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mibolerone from Androgen receptor (unknown origin) measured by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to bicalutamide-resistant Androgen receptor T878A mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Binding affinity to rat Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Binding affinity to human BRD3 BD2 (306 to 417 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to human Androgen receptor measured by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity to human BRD2 BD2 (349 to 460 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to Androgen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to human BRD4 BD2 (333 to 460 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to human Androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]DHT from Androgen receptor expressed in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Binding affinity to human BRD4 BD1 (44 to 168 residues) by fluorescence polarization assayMore data for this Ligand-Target Pair