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Found 157 with Last Name = 'yamaotsu' and Initial = 'n'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50013388(6-Ethyl-3-(1-hydroxy-cyclopropylmethyl)-11,11-dime...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50321030(CHEMBL1163924 | N-{[(1R,9R,10S,13R)-17-(cyclopropy...)
Affinity DataKi:  0.135nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50321028((1S,2R,6S,14R,15R,16R)-3-(cyclopropylmethyl)-11,15...)
Affinity DataKi:  0.152nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50049805(CHEMBL169703 | Thiophene-3-carboxylic acid [5-(2-f...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50274257((2E)-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-...)
Affinity DataKi:  0.195nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50274257((2E)-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-...)
Affinity DataKi:  0.225nMAssay Description:Displacement of [3H]U69593 from guinea pig cerebellum kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50321029((1R,2R,6S,14R,15R,16S)-3-(cyclopropylmethyl)-11,15...)
Affinity DataKi:  0.279nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50274257((2E)-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-...)
Affinity DataKi:  0.582nMAssay Description:Displacement of [3H]DAMGO from guinea pig forebrain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]DPDPE from mouse whole brain DORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50159165((2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028063(CHEMBL3338874)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50321024((1R,2S,4R,5S)-dimethyl 3,7-dimethyl-9-oxo-2,4-di(p...)
Affinity DataKi:  15nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028063(CHEMBL3338874)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  33.7nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50321031(CHEMBL1164183 | Tyr-c[D-cys-Phe-D-Cys]-NH2)
Affinity DataKi:  38.7nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50321032((2S,5S)-2-(4-methoxyphenyl)-5-methyl-1-(3-phenylpr...)
Affinity DataKi:  39nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028063(CHEMBL3338874)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]DPDPE from mouse whole brain DORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028060(CHEMBL3338872)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028061(CHEMBL3338873)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028064(CHEMBL3338875)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028065(CHEMBL3338876)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028069(CHEMBL3338877)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028071(CHEMBL3338878)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028072(CHEMBL3338879)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028073(CHEMBL3338880)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028077(CHEMBL3338881)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028078(CHEMBL3338882)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69593 from guinea pig cerebellum KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028079(CHEMBL3338867)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028081(CHEMBL3338868)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028082(CHEMBL3338869)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028084(CHEMBL3338870)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028085(CHEMBL3338871)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028060(CHEMBL3338872)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028061(CHEMBL3338873)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028064(CHEMBL3338875)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028065(CHEMBL3338876)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028069(CHEMBL3338877)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028071(CHEMBL3338878)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028072(CHEMBL3338879)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028073(CHEMBL3338880)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028077(CHEMBL3338881)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028078(CHEMBL3338882)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028086(CHEMBL3338883)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028087(CHEMBL3338884)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from mouse whole brain DORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50028079(CHEMBL3338867)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from mouse whole brain DORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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