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Found 60 with Last Name = 'yang' and Initial = 'jh'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant MAOB assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50260171(CHEMBL4062286)
Affinity DataIC50:  144nMAssay Description:Inhibition of human recombinant MAOB assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219240(4-[4-(benzyloxy)piperidino]butyl-N-(4-chlorophenyl...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219232(4-[4-(benzhydryloxy)piperidino]butyl-4-chlorobenzo...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219230(4-[4-(benzyloxy)piperidino]butyl-4-fluorobenzoate ...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219235(4-[4-(benzyloxy)piperidino]butyl-N-(4-fluorophenyl...)
Affinity DataIC50:  780nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219245(4-[4-(benzhydryloxy)piperidino]butyl 4-fluorobenzo...)
Affinity DataIC50:  840nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataIC50:  960nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) assessed as N-methyldihydronicotinamide oxidation per mg of protein a...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50553951(CHEMBL4782189)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human PMA-differentiated THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219238(4-[4-(benzhydryloxy)piperidino]butyl benzoate | CH...)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219233(4-[4-(benzyloxy)piperidino]butyl-3-chlorobenzoate ...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219231(4-[4-(benzyloxy)piperidino]butyl-3-fluorobenzoate ...)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219248(4-[4-(benzyloxy)piperidino]butyl benzoate | CHEMBL...)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219249(4-[4-(benzhydryloxy)piperidino]butyl-4-(tert-butyl...)
Affinity DataIC50:  2.41E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219241(4-[4-(benzhydryloxy)piperidino]butyl-N-(4-fluoroph...)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219242(4-[4-(benzhydryloxy)piperidino]butyl-N-(4-chloroph...)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219234(4-[4-(benzhydryloxy)piperidino]butyl 3-chlorobenzo...)
Affinity DataIC50:  3.39E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219244(4-[4-(benzyloxy)piperidino]butyl-4-chlorobenzoate ...)
Affinity DataIC50:  3.52E+3nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50339150(5,7-dihydroxy-2-(4-hydroxyphenyl)-3-((2R,3S,4S,5S,...)
Affinity DataIC50:  3.84E+3nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) assessed as N-methyldihydronicotinamide oxidation per mg of protein a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219239(4-[4-(benzhydryloxy)piperidino]butyl 4-isopropylbe...)
Affinity DataIC50:  3.89E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219236(4-[4-(benzyloxy)piperidino]butyl-4-nitrobenzoate |...)
Affinity DataIC50:  5.23E+3nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  6.56E+3nMAssay Description:Inhibition of human recombinant MAOA assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219237(4-[4-(benzhydryloxy)piperidino]butyl-4-nitrobenzoa...)
Affinity DataIC50:  7.25E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  7.54E+3nMAssay Description:Inhibition of human recombinant MAOB assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219246(4-[4-(benzhydryloxy)piperidino]butyl 3-fluorobenzo...)
Affinity DataIC50:  7.72E+3nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219229(4-[4-(benzyloxy)piperidino]butyl-4-isopropylbenzoa...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219247(4-[4-(benzyloxy)piperidino]butyl-4-(tert-butyl)-be...)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219242(4-[4-(benzhydryloxy)piperidino]butyl-N-(4-chloroph...)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219229(4-[4-(benzyloxy)piperidino]butyl-4-isopropylbenzoa...)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of Electrophorus electricus AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219247(4-[4-(benzyloxy)piperidino]butyl-4-(tert-butyl)-be...)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219241(4-[4-(benzhydryloxy)piperidino]butyl-N-(4-fluoroph...)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219245(4-[4-(benzhydryloxy)piperidino]butyl 4-fluorobenzo...)
Affinity DataIC50:  2.22E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219239(4-[4-(benzhydryloxy)piperidino]butyl 4-isopropylbe...)
Affinity DataIC50:  2.32E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50:  2.42E+4nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human PMA-differentiated THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50339149(CHEMBL1689259 | beta-(3,4-dihydroxyphenyl)ethyl-3-...)
Affinity DataIC50:  2.68E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219237(4-[4-(benzhydryloxy)piperidino]butyl-4-nitrobenzoa...)
Affinity DataIC50:  2.68E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50339147(CHEMBL1689257 | beta-(4-hydroxyphenyl)ethyl-4-O-E-...)
Affinity DataIC50:  3.07E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219238(4-[4-(benzhydryloxy)piperidino]butyl benzoate | CH...)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219246(4-[4-(benzhydryloxy)piperidino]butyl 3-fluorobenzo...)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50339148(CHEMBL1689258 | beta-(3,4-dihydroxyphenyl)ethyl-6-...)
Affinity DataIC50:  3.23E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50269516(CHEMBL518414 | Calceolarioside B)
Affinity DataIC50:  3.53E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219232(4-[4-(benzhydryloxy)piperidino]butyl-4-chlorobenzo...)
Affinity DataIC50:  3.84E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Mus musculus (Mouse))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50342164(5-(3-Chlorobenzyloxy)benzene-1,3-diol | CHEMBL1766...)
Affinity DataIC50:  5.47E+4nMAssay Description:Inhibition of tyrosinase activity in alpha-MSH-stimulated mouse B16 cells using L-tyrosine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219234(4-[4-(benzhydryloxy)piperidino]butyl 3-chlorobenzo...)
Affinity DataIC50:  5.79E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosinase(Mus musculus (Mouse))
Catholic University Of Daegu

Curated by ChEMBL
LigandPNGBDBM50342165(5-(3,4-Dichlorobenzyloxy)benzene-1,3-diol | CHEMBL...)
Affinity DataIC50:  6.64E+4nMAssay Description:Inhibition of tyrosinase activity in alpha-MSH-stimulated mouse B16 cells using L-tyrosine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  6.73E+4nMAssay Description:Displacement of [3H]R-1881 from Androgen receptor of LNCaP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Woosuk University

Curated by ChEMBL
LigandPNGBDBM50219249(4-[4-(benzhydryloxy)piperidino]butyl-4-(tert-butyl...)
Affinity DataIC50:  7.89E+4nMAssay Description:Inhibition of human BChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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