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Found 369 with Last Name = 'young' and Initial = 'lc'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206172(1-(benzo[d][1,3]dioxol-5-ylmethyl)-2,3,4,9-tetrahy...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206189(1-(2-(propylthio)benzyl)-2,3,4,9-tetrahydro-1H-pyr...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206163(1-(3-Methoxy-benzyl)-2,3,4,9-tetrahydro-1H-beta-ca...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206164(1-(2-(methylthio)benzyl)-2,3,4,9-tetrahydro-1H-pyr...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206169(1-(benzo[d][1,3]dioxol-5-ylmethyl)-6-methoxy-2,3,4...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206175(1-(3-methoxybenzyl)-6-methoxy-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206186(2-fluoro-6-((2,3,4,9-tetrahydro-1H-pyrido[3,4-b]in...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257823(CHEMBL4089551)
Affinity DataKi:  80nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206168(2,9-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibe...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]DPCPX from human cloned adenosine A1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257884(CHEMBL4065551)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206178((E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279446(8-[3-(2-Diethylaminoethoxy)phenyl]-1,3-dimethylxan...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206183((E)-6-((benzyl(methyl)amino)methyleneamino)-2,3-di...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279444(1,3-Dimethyl-8-[4-methoxy-3-(2-morpholin-4-ylethox...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206161(1-(4-(methylthio)benzyl)-2,3,4,9-tetrahydro-1H-pyr...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206174((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206173((E)-7-((3,4-dihydroisoquinolin-2(1H)-yl)methylenea...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206190((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206165((E)-7-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206162((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257927(CHEMBL4061406)
Affinity DataKi:  300nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206162((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206184((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206192((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206177((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257824(CHEMBL4074174)
Affinity DataKi:  400nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206165((E)-7-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279464(1,3-Dimethyl-8-[3-(2-pyrrolidin-1-ylethoxy)-phenyl...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279422(8-[3-(2-Dimethylaminoethoxy)-4-methoxyphenyl]-1,3-...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279445(8-[3-(2-Dimethylaminoethoxy)phenyl]-1,3-dimethylxa...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206192((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206190((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]DPCPX from human cloned adenosine A1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279423(8-[3-(2-Diethylaminoethoxy)-4-methoxyphenyl]-1,3-d...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279730(8-[4-(2-Dimethylaminoethoxy)-3-methoxyphenyl]-1,3-...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257859(CHEMBL4096206)
Affinity DataKi:  610nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257822(CHEMBL4088616)
Affinity DataKi:  650nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279732(1,3-Dimethyl-8-[3-methoxy-4-(2-piperidin-1-ylethox...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206184((E)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257925(CHEMBL4086169)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206170(1-(3-methoxyphenyl)-4,9-dihydro-3H-pyrido[3,4-b]in...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279447(1,3-Dimethyl-8-[3-(2-piperidin-4-ylethoxy)phenyl]x...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279445(8-[3-(2-Dimethylaminoethoxy)phenyl]-1,3-dimethylxa...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]DPCPX from human cloned adenosine A1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206177((E)-3-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257823(CHEMBL4089551)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50279421(1,3-Dimethyl-8-[3-methoxy-4-(2-pyrrolidin-4-yletho...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]ZM-241385 from human cloned adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206174((E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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