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27 similar compounds to monomer 50185261

Compile data set for download or QSAR
Wt: 459.4
BDBM50005459
Wt: 410.9
BDBM50008166
Wt: 459.4
BDBM50008170
Wt: 434.9
BDBM50008176
Wt: 382.8
BDBM50008181
Wt: 403.3
BDBM50008182
Wt: 368.8
BDBM50008184
Wt: 394.8
BDBM50008186
Wt: 368.8
BDBM50008188
Wt: 354.8
BDBM50008189
Wt: 403.3
BDBM50008191
Wt: 389.2
BDBM50008195
Wt: 382.8
BDBM50008196
Wt: 340.8
BDBM50008199
Wt: 354.8
BDBM50008200
Displayed 1 to 15 (of 27 total )  |  Next  |  Last  >>

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 46 hits for monomerid = 50005459,50008166,50008170,50008176,50008181,50008182,50008184,50008186,50008188,50008189,50008191,50008195,50008196,50008199,50008200   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cholecystokinin B


(GUINEA PIG)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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22n/an/an/an/an/an/an/an/a



Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database




Eur J Pharmacol 162: 273-80 (1989)


Article DOI: 10.1016/0014-2999(89)90290-2
BindingDB Entry DOI: 10.7270/Q2QF8RB7
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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49n/an/an/an/an/an/an/an/a



Center for Bio-Pharmaceutical Sciences

Curated by ChEMBL


Assay Description
Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranes


J Med Chem 35: 1042-9 (1992)


Article DOI: 10.1021/jm00084a009
BindingDB Entry DOI: 10.7270/Q2HT2N8R
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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129n/an/an/an/an/an/an/an/a



Universitá di Siena

Curated by ChEMBL


Assay Description
Binding affinity against Cholecystokinin type A receptor using [125I]-(BH)-CCK-8 as radioligand in rat pancreas.


J Med Chem 39: 860-72 (1996)


Article DOI: 10.1021/jm950423p
BindingDB Entry DOI: 10.7270/Q2222SVD
More data for this
Ligand-Target Pair
Cholecystokinin B


(GUINEA PIG)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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1.90E+3n/an/an/an/an/an/an/an/a



Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database




Eur J Pharmacol 162: 273-80 (1989)


Article DOI: 10.1016/0014-2999(89)90290-2
BindingDB Entry DOI: 10.7270/Q2QF8RB7
More data for this
Ligand-Target Pair
Cholecystokinin B


(GUINEA PIG)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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2.20E+3n/an/an/an/an/an/an/an/a



Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database




Eur J Pharmacol 162: 273-80 (1989)


Article DOI: 10.1016/0014-2999(89)90290-2
BindingDB Entry DOI: 10.7270/Q2QF8RB7
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 50n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic acini


Bioorg Med Chem Lett 3: 861-866 (1993)


Article DOI: 10.1016/S0960-894X(00)80681-2
BindingDB Entry DOI: 10.7270/Q2J103M7
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 50n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreas


Bioorg Med Chem Lett 3: 889-894 (1993)


Article DOI: 10.1016/S0960-894X(00)80687-3
BindingDB Entry DOI: 10.7270/Q28G8M63
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(MOUSE)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 3.00E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortex


Bioorg Med Chem Lett 3: 889-894 (1993)


Article DOI: 10.1016/S0960-894X(00)80687-3
BindingDB Entry DOI: 10.7270/Q28G8M63
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008166
PNG
(4-(3-Chloro-benzoylamino)-4-(3,3-diethyl-pentylcar...)
Show SMILES CCC(CC)(CC)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C21H31ClN2O4/c1-4-21(5-2,6-3)12-13-23-20(28)17(10-11-18(25)26)24-19(27)15-8-7-9-16(22)14-15/h7-9,14,17H,4-6,10-13H2,1-3H3,(H,23,28)(H,24,27)(H,25,26)
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n/an/a 900n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(Homo sapiens (Human))
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 2.50E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to cholecystokinin type B receptor in rabbit gastric gland


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008176
PNG
(4-(3-Chloro-benzoylamino)-4-(spiro[5.5]undec-3-ylc...)
Show SMILES OC(=O)CCC(NC(=O)c1cccc(Cl)c1)C(=O)NC1CCC2(CCCCC2)CC1
Show InChI InChI=1S/C23H31ClN2O4/c24-17-6-4-5-16(15-17)21(29)26-19(7-8-20(27)28)22(30)25-18-9-13-23(14-10-18)11-2-1-3-12-23/h4-6,15,18-19H,1-3,7-14H2,(H,25,30)(H,26,29)(H,27,28)
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n/an/a 7.80E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 50n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008181
PNG
(4-(3-Chloro-benzoylamino)-4-(4,4-dimethyl-pentylca...)
Show SMILES CC(C)(C)CCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C19H27ClN2O4/c1-19(2,3)10-5-11-21-18(26)15(8-9-16(23)24)22-17(25)13-6-4-7-14(20)12-13/h4,6-7,12,15H,5,8-11H2,1-3H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a 3.20E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008182
PNG
(4-(2,3-Dichloro-benzoylamino)-4-(3,3-dimethyl-buty...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1Cl
Show InChI InChI=1S/C18H24Cl2N2O4/c1-18(2,3)9-10-21-17(26)13(7-8-14(23)24)22-16(25)11-5-4-6-12(19)15(11)20/h4-6,13H,7-10H2,1-3H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a 2.90E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008186
PNG
(4-(3-Chloro-benzoylamino)-4-(4,4-dimethyl-cyclohex...)
Show SMILES CC1(C)CCC(CC1)NC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C20H27ClN2O4/c1-20(2)10-8-15(9-11-20)22-19(27)16(6-7-17(24)25)23-18(26)13-4-3-5-14(21)12-13/h3-5,12,15-16H,6-11H2,1-2H3,(H,22,27)(H,23,26)(H,24,25)
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n/an/a 5.80E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008188
PNG
(4-(3-Chloro-benzoylamino)-4-hexylcarbamoyl-butyric...)
Show SMILES CCCCCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C18H25ClN2O4/c1-2-3-4-5-11-20-18(25)15(9-10-16(22)23)21-17(24)13-7-6-8-14(19)12-13/h6-8,12,15H,2-5,9-11H2,1H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 2.15E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008189
PNG
(4-(3-Chloro-benzoylamino)-4-(3-methyl-butylcarbamo...)
Show SMILES CC(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C17H23ClN2O4/c1-11(2)8-9-19-17(24)14(6-7-15(21)22)20-16(23)12-4-3-5-13(18)10-12/h3-5,10-11,14H,6-9H2,1-2H3,(H,19,24)(H,20,23)(H,21,22)
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n/an/a>1.00E+5n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of [125I](BH)-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic acini; Inactive


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin A receptor


(Cavia porcellus)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 66n/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Compound was evaluated for the binding affinity against Cholecystokinin type A receptor in cortical cells.


J Med Chem 32: 739-42 (1989)


Article DOI: 10.1021/jm00124a003
BindingDB Entry DOI: 10.7270/Q2M61J8V
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008195
PNG
(4-(3,4-Dichloro-benzoylamino)-4-pentylcarbamoyl-bu...)
Show SMILES CCCCCNC(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C17H22Cl2N2O4/c1-2-3-4-9-20-17(25)14(7-8-15(22)23)21-16(24)11-5-6-12(18)13(19)10-11/h5-6,10,14H,2-4,7-9H2,1H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 1.02E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% the specific binding of [125I](BH)-CCK-8 to CCK-B(B2) in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008196
PNG
(4-(3-Chloro-benzoylamino)-4-heptylcarbamoyl-butyri...)
Show SMILES CCCCCCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C19H27ClN2O4/c1-2-3-4-5-6-12-21-19(26)16(10-11-17(23)24)22-18(25)14-8-7-9-15(20)13-14/h7-9,13,16H,2-6,10-12H2,1H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a 2.80E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008166
PNG
(4-(3-Chloro-benzoylamino)-4-(3,3-diethyl-pentylcar...)
Show SMILES CCC(CC)(CC)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C21H31ClN2O4/c1-4-21(5-2,6-3)12-13-23-20(28)17(10-11-18(25)26)24-19(27)15-8-7-9-16(22)14-15/h7-9,14,17H,4-6,10-13H2,1-3H3,(H,23,28)(H,24,27)(H,25,26)
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n/an/a 8.00E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008186
PNG
(4-(3-Chloro-benzoylamino)-4-(4,4-dimethyl-cyclohex...)
Show SMILES CC1(C)CCC(CC1)NC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C20H27ClN2O4/c1-20(2)10-8-15(9-11-20)22-19(27)16(6-7-17(24)25)23-18(26)13-4-3-5-14(21)12-13/h3-5,12,15-16H,6-11H2,1-2H3,(H,22,27)(H,23,26)(H,24,25)
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n/an/a>1.00E+5n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of [125I](BH)-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic acini; Inactive


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008199
PNG
(4-Butylcarbamoyl-4-(3-chloro-benzoylamino)-butyric...)
Show SMILES CCCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C16H21ClN2O4/c1-2-3-9-18-16(23)13(7-8-14(20)21)19-15(22)11-5-4-6-12(17)10-11/h4-6,10,13H,2-3,7-9H2,1H3,(H,18,23)(H,19,22)(H,20,21)
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n/an/a 5.06E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008191
PNG
(4-(3,4-Dichloro-benzoylamino)-4-(3,3-dimethyl-buty...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C18H24Cl2N2O4/c1-18(2,3)8-9-21-17(26)14(6-7-15(23)24)22-16(25)11-4-5-12(19)13(20)10-11/h4-5,10,14H,6-9H2,1-3H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a 3.10E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008200
PNG
(4-(4-Chloro-benzoylamino)-4-pentylcarbamoyl-butyri...)
Show SMILES CCCCCNC(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)cc1
Show InChI InChI=1S/C17H23ClN2O4/c1-2-3-4-11-19-17(24)14(9-10-15(21)22)20-16(23)12-5-7-13(18)8-6-12/h5-8,14H,2-4,9-11H2,1H3,(H,19,24)(H,20,23)(H,21,22)
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n/an/a 3.13E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008182
PNG
(4-(2,3-Dichloro-benzoylamino)-4-(3,3-dimethyl-buty...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1Cl
Show InChI InChI=1S/C18H24Cl2N2O4/c1-18(2,3)9-10-21-17(26)13(7-8-14(23)24)22-16(25)11-5-4-6-12(19)15(11)20/h4-6,13H,7-10H2,1-3H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a>1.00E+5n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of [125I](BH)-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic acini; Inactive


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008195
PNG
(4-(3,4-Dichloro-benzoylamino)-4-pentylcarbamoyl-bu...)
Show SMILES CCCCCNC(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C17H22Cl2N2O4/c1-2-3-4-9-20-17(25)14(7-8-15(22)23)21-16(24)11-5-6-12(18)13(19)10-11/h5-6,10,14H,2-4,7-9H2,1H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 8.60E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(Homo sapiens (Human))
BDBM50008184
PNG
(4-(3-Chloro-benzoylamino)-4-(3,3-dimethyl-butylcar...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C18H25ClN2O4/c1-18(2,3)9-10-20-17(25)14(7-8-15(22)23)21-16(24)12-5-4-6-13(19)11-12/h4-6,11,14H,7-10H2,1-3H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 2.20E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% the specific binding of [3H]pentagastrin to Cholecystokinin type B receptor in rabbit gastric gland


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008184
PNG
(4-(3-Chloro-benzoylamino)-4-(3,3-dimethyl-butylcar...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C18H25ClN2O4/c1-18(2,3)9-10-20-17(25)14(7-8-15(22)23)21-16(24)12-5-4-6-13(19)11-12/h4-6,11,14H,7-10H2,1-3H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 1.01E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008199
PNG
(4-Butylcarbamoyl-4-(3-chloro-benzoylamino)-butyric...)
Show SMILES CCCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C16H21ClN2O4/c1-2-3-9-18-16(23)13(7-8-14(20)21)19-15(22)11-5-4-6-12(17)10-11/h4-6,10,13H,2-3,7-9H2,1H3,(H,18,23)(H,19,22)(H,20,21)
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n/an/a>1.00E+5n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of [125I](BH)-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic acini; Inactive


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008196
PNG
(4-(3-Chloro-benzoylamino)-4-heptylcarbamoyl-butyri...)
Show SMILES CCCCCCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C19H27ClN2O4/c1-2-3-4-5-6-12-21-19(26)16(10-11-17(23)24)22-18(25)14-8-7-9-15(20)13-14/h7-9,13,16H,2-6,10-12H2,1H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a>1.00E+5n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of [125I](BH)-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic acini; Inactive


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008189
PNG
(4-(3-Chloro-benzoylamino)-4-(3-methyl-butylcarbamo...)
Show SMILES CC(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C17H23ClN2O4/c1-11(2)8-9-19-17(24)14(6-7-15(21)22)20-16(23)12-4-3-5-13(18)10-12/h3-5,10-11,14H,6-9H2,1-2H3,(H,19,24)(H,20,23)(H,21,22)
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n/an/a 3.53E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008188
PNG
(4-(3-Chloro-benzoylamino)-4-hexylcarbamoyl-butyric...)
Show SMILES CCCCCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C18H25ClN2O4/c1-2-3-4-5-11-20-18(25)15(9-10-16(22)23)21-17(24)13-7-6-8-14(19)12-13/h6-8,12,15H,2-5,9-11H2,1H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 8.00E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008184
PNG
(4-(3-Chloro-benzoylamino)-4-(3,3-dimethyl-butylcar...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C18H25ClN2O4/c1-18(2,3)9-10-20-17(25)14(7-8-15(22)23)21-16(24)12-5-4-6-13(19)11-12/h4-6,11,14H,7-10H2,1-3H3,(H,20,25)(H,21,24)(H,22,23)
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n/an/a 9.05E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008200
PNG
(4-(4-Chloro-benzoylamino)-4-pentylcarbamoyl-butyri...)
Show SMILES CCCCCNC(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)cc1
Show InChI InChI=1S/C17H23ClN2O4/c1-2-3-4-11-19-17(24)14(9-10-15(21)22)20-16(23)12-5-7-13(18)8-6-12/h5-8,14H,2-4,9-11H2,1H3,(H,19,24)(H,20,23)(H,21,22)
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n/an/a 3.62E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008176
PNG
(4-(3-Chloro-benzoylamino)-4-(spiro[5.5]undec-3-ylc...)
Show SMILES OC(=O)CCC(NC(=O)c1cccc(Cl)c1)C(=O)NC1CCC2(CCCCC2)CC1
Show InChI InChI=1S/C23H31ClN2O4/c24-17-6-4-5-16(15-17)21(29)26-19(7-8-20(27)28)22(30)25-18-9-13-23(14-10-18)11-2-1-3-12-23/h4-6,15,18-19H,1-3,7-14H2,(H,25,30)(H,26,29)(H,27,28)
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n/an/a 3.50E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008181
PNG
(4-(3-Chloro-benzoylamino)-4-(4,4-dimethyl-pentylca...)
Show SMILES CC(C)(C)CCCNC(=O)C(CCC(O)=O)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C19H27ClN2O4/c1-19(2,3)10-5-11-21-18(26)15(8-9-16(23)24)22-17(25)13-6-4-7-14(20)12-13/h4,6-7,12,15H,5,8-11H2,1-3H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a 2.79E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
CCKBR


(RAT)
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 3.00E+3n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Inhibition of the specific binding of [125I](BH)-CCK-8 to Cholecystokinin type B receptor in rat brain cortex


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 18n/an/an/an/an/an/a



Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of binding of [125I]- CCK-33 to rat pancreas


J Med Chem 33: 591-5 (1990)


Article DOI: 10.1021/jm00164a020
BindingDB Entry DOI: 10.7270/Q29K4BTP
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(Homo sapiens (Human))
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 1.90E+3n/an/an/an/an/an/a



Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of binding of [125I]gastrin to Cholecystokinin type B receptor from guinea pig gastric glands


J Med Chem 33: 591-5 (1990)


Article DOI: 10.1021/jm00164a020
BindingDB Entry DOI: 10.7270/Q29K4BTP
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(Homo sapiens (Human))
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 5.60E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortex


Bioorg Med Chem Lett 3: 861-866 (1993)


Article DOI: 10.1016/S0960-894X(00)80681-2
BindingDB Entry DOI: 10.7270/Q2J103M7
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 22n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Displacement of [125I]-CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assay


Bioorg Med Chem Lett 2: 1251-1256 (1992)


Article DOI: 10.1016/S0960-894X(00)80224-3
BindingDB Entry DOI: 10.7270/Q24T6J92
More data for this
Ligand-Target Pair
Cholecystokinin A receptor


(Cavia porcellus)
BDBM50008170
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)
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n/an/a 2.20E+3n/an/an/an/an/an/a



Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of binding of [125I]- CCK-33 to guinea pig cortex


J Med Chem 33: 591-5 (1990)


Article DOI: 10.1021/jm00164a020
BindingDB Entry DOI: 10.7270/Q29K4BTP
More data for this
Ligand-Target Pair
Cholecystokinin A receptor


(Cavia porcellus)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 1.24E+4n/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Compound was evaluated for the binding affinity against CCK A receptor in cortical cells.


J Med Chem 32: 739-42 (1989)


Article DOI: 10.1021/jm00124a003
BindingDB Entry DOI: 10.7270/Q2M61J8V
More data for this
Ligand-Target Pair
Cholecystokinin A receptor


(Cavia porcellus)
BDBM50005459
PNG
(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Show SMILES CCCCCN(CCCCC)C(=O)[C@@H](CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C22H32Cl2N2O4/c1-3-5-7-13-26(14-8-6-4-2)22(30)19(11-12-20(27)28)25-21(29)16-9-10-17(23)18(24)15-16/h9-10,15,19H,3-8,11-14H2,1-2H3,(H,25,29)(H,27,28)/t19-/m1/s1
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n/an/a 66n/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Inhibition of [125I]-Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreatic membranes.


J Med Chem 34: 3350-9 (1992)


Article DOI: 10.1021/jm00116a002
BindingDB Entry DOI: 10.7270/Q2M907M8
More data for this
Ligand-Target Pair
Cholecystokinin receptor


(RAT)
BDBM50008191
PNG
(4-(3,4-Dichloro-benzoylamino)-4-(3,3-dimethyl-buty...)
Show SMILES CC(C)(C)CCNC(=O)C(CCC(O)=O)NC(=O)c1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C18H24Cl2N2O4/c1-18(2,3)8-9-21-17(26)14(6-7-15(23)24)22-16(25)11-4-5-12(19)13(20)10-11/h4-5,10,14H,6-9H2,1-3H3,(H,21,26)(H,22,25)(H,23,24)
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n/an/a 1.88E+4n/an/an/an/an/an/a



Rotta Research Laboratorium

Curated by ChEMBL


Assay Description
Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic acini


J Med Chem 35: 28-38 (1992)


Article DOI: 10.1021/jm00079a003
BindingDB Entry DOI: 10.7270/Q2XS5W11
More data for this
Ligand-Target Pair