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Found 36 Enz. Inhib. hit(s) with Target = 'Protein ADM2'
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570409(CHEMBL4857810)
Affinity DataIC50:  0.631nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570410(CHEMBL4851152)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570411(CHEMBL4877585)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570413(CHEMBL4850259)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570396(CHEMBL4871934)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570397(CHEMBL4852669)
Affinity DataIC50:  7.90nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50246690(Ac-WVTHRLAGLLSRSGGVVRKNFVPTDVGPFAF-NH2 | CHEMBL503...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570401(CHEMBL4879142)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570400(CHEMBL4876643)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570402(CHEMBL4856402)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570408(CHEMBL4873687)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50246693(Ac-WVTH[Cit]LAGLLS[Cit]SGGVVRKNFVPTDVGPFAF-NH2 | C...)
Affinity DataIC50:  108nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570404(CHEMBL4850583)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570398(CHEMBL4861626)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570388(CHEMBL4858139)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50000743(CHEMBL525571 | [Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Se...)
Affinity DataIC50:  266nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570394(CHEMBL4866548)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570395(CHEMBL4866915)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50246697(Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGPFAF-NH...)
Affinity DataIC50:  318nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50246708(Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGP[1-Nal...)
Affinity DataIC50:  375nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50246709(Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGP[2-Nal...)
Affinity DataIC50:  418nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50025073(CHEMBL2372187)
Affinity DataIC50:  496nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570406(CHEMBL4862324)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570412(CHEMBL4853766)
Affinity DataIC50:  794nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570390(CHEMBL4851106)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570405(CHEMBL4874859)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570393(CHEMBL4878394)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570386(CHEMBL4864804)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570403(CHEMBL4874651)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570407(CHEMBL4865654)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50025076(CHEMBL2372194)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570399(CHEMBL4846989)
Affinity DataIC50:  3.16E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570392(CHEMBL4870543)
Affinity DataIC50:  7.94E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570389(CHEMBL4867733)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570387(CHEMBL4853613)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ADM2(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50570391(CHEMBL4876213)
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed