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Found 20 Enz. Inhib. hit(s) with Target = 'BRCA1-associated RING domain protein 1'
TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM63209(3-(1-phenyl-2-thioxo-2,3-dihydro-1H-imidazol-4-yl)...)
Affinity DataIC50:  3.53nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48281((2-fluorophenyl)-[5-[1-(2-methoxyethyl)-2,5-dimeth...)
Affinity DataIC50:  493nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79631(5'-methoxy-1'-methyl-5H-spiro[benzimidazo[...)
Affinity DataIC50:  1.18E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM65180((3,4-Dihydro-2H-quinolin-1-yl)-acetic acid [1-(2-h...)
Affinity DataIC50:  1.97E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79632(2-hydroxy-6-isopropyl-cyclohepta-2,4,6-trien-1-one...)
Affinity DataIC50:  3.89E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM72275((E)-2-butenedioic acid O4-[2-[(diphenylmethyl)amin...)
Affinity DataIC50:  3.90E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79636(1-(2-furanylmethyl)-2-imino-10-methyl-5-oxo-N-(2-p...)
Affinity DataIC50:  4.13E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM60287(2-nitro-N-(8-quinolinyl)benzenesulfonamide | 2-nit...)
Affinity DataIC50:  4.37E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79637(5-(4-acetylphenyl)-N-(4-pyridin-2-yl-1,3-thiazol-2...)
Affinity DataIC50:  4.85E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM41443(MLS000060380 | N-(2,5-diethoxy-4-morpholin-4-yl-ph...)
Affinity DataIC50:  5.07E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM58130((6E)-6-[4-[N'-[(1E)-1-(6-ketocyclohexa-2,4-dien-1-...)
Affinity DataIC50:  5.35E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48124((4,8-dimethylquinazolin-2-yl)-[3-(3-morpholinoprop...)
Affinity DataIC50:  5.59E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79634((E)-3-(2-Chloro-6-fluoro-phenyl)-1-(4-hydroxy-phen...)
Affinity DataIC50:  6.64E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79633(4-[2-(4,5-dichloro-6-keto-pyridazin-1-yl)acetyl]-3...)
Affinity DataIC50:  8.39E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM43474((3Z,5E)-1-ethyl-3,5-bis(3-hydroxy-4-methoxy-benzyl...)
Affinity DataIC50:  9.78E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM61625(2-chloranyl-N-[2-[(2-chloranylpyridin-3-yl)carbony...)
Affinity DataIC50:  1.01E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79083(2-[2-(4-methoxyphenyl)-7-methyl-4-oxidanylidene-py...)
Affinity DataIC50:  1.06E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM70514(2-[(1-methyl-3-nitro-1H-1,2,4-triazol-5-yl)thio]-5...)
Affinity DataIC50:  1.23E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79630(MLS000049666 | N-[4-[5-(3,4,5-trimethoxyphenyl)-1,...)
Affinity DataIC50:  1.34E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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TargetBRCA1-associated RING domain protein 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79635(4-[(4-amino-6,7-dimethoxy-2-quinazolinyl)amino]ben...)
Affinity DataIC50:  1.43E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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