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Found 55 Enz. Inhib. hit(s) with Target = 'Bis(5'-adenosyl)-triphosphatase'
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350516(CHEMBL1812066)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350512(CHEMBL1812070)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350513(CHEMBL1812069)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81576(AppppA analog, 6 (X=S))
Affinity DataKi:  35nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350514(CHEMBL1812068)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50350515(CHEMBL1812067)
Affinity DataKi:  35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81584(AppppA analog, 12 (X=S))
Affinity DataKi:  40nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81586(AppppA analog, 13 (X=S))
Affinity DataKi:  65nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81590(AppppA analog, 15 (X=S))
Affinity DataKi:  78nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81593(AppppA analog, 17 (X=S))
Affinity DataKi:  110nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81575(AppppA analog, 5 (X=S))
Affinity DataKi:  220nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81580(AppppA analog, 9 (X=S))
Affinity DataKi:  230nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81592(AppppA analog, 17 (X=O))
Affinity DataKi:  420nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81588(AppppA analog, 14 (X=S))
Affinity DataKi:  700nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81587(AppppA analog, 14 (X=O))
Affinity DataKi:  900nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81574(AppppA analog, 5 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81583(AppppA analog, 12 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81589(AppppA analog, 15 (X=O))
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81570(AppppA analog, 1 (X=O))
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81571(AppppA analog, 2 (X=S))
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81591(AppppA analog, 16 (X=S))
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81579(AppppA analog, 8 (X=S))
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81585(AppppA analog, 13 (X=O))
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81581(AppppA analog, 10 (X=S))
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81577(AppppA analog, 6 (X=O))
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81582(AppppA analog, 11 (X=S))
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81578(AppppA analog, 7 (X=S))
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81572(AppppA analog, 3 (X=S))
Affinity DataKi:  8.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM81573(AppppA analog, 4 (X=S))
Affinity DataKi:  8.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580671(CHEMBL5083166)
Affinity DataIC50:  49nMAssay Description:Inhibition of human FHIT expressed in Escherichia coli BL21(DE3)-RIL cells using AP3A as substrate pretreated for 10 mins followed by substrate addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580669(CHEMBL5079345)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580669(CHEMBL5079345)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580665(CHEMBL5078809)
Affinity DataIC50:  140nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580675(CHEMBL5075611)
Affinity DataIC50:  770nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580679(CHEMBL5093727)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580672(CHEMBL5078205)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580665(CHEMBL5078809)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580667(CHEMBL5069986)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580674(CHEMBL5076149)
Affinity DataIC50:  3.43E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580676(CHEMBL5081769)
Affinity DataIC50:  3.73E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580677(CHEMBL5075193)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580659(CHEMBL5088775)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580678(CHEMBL5093738)
Affinity DataIC50:  4.24E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580673(CHEMBL1520857)
Affinity DataIC50:  4.66E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580668(CHEMBL1444825)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580664(CHEMBL5077048)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580670(CHEMBL5092878)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580663(CHEMBL5083554)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580671(CHEMBL5083166)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50580666(CHEMBL5081492)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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