TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human GRK4 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 69.9nMAssay Description:Inhibition of human GRK4 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of human GRK4 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of human GRK4 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human GRK4 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of GRK4-mediated bovine tubulin phosphorylation by scintillation countingMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of full-length recombinant human GST-tagged GRK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of full-length recombinant human GST-tagged GRK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged GRK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length GST-tagged GRK4 expressed in baculovirus expression systemMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human GRK4 using casein as substrateMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of full-length recombinant human GST-tagged GRK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.47E+4nMAssay Description:Inhibition of Protein kinase C deltaMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 17nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 37nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 2.90E+3nMAssay Description:Binding affinity to GRK4More data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 590nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 4.20E+3nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 97nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 6.20E+3nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 2.80E+3nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 4(Homo sapiens (Human))
Ontario Institute For Cancer Research
Curated by ChEMBL
Ontario Institute For Cancer Research
Curated by ChEMBL
Affinity DataKd: 2.30E+3nMAssay Description:Binding constant for GRK4 kinase domainMore data for this Ligand-Target Pair