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Found 158 Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor 52'
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556717(CHEMBL4780703)
Affinity DataIC50:  630nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556698(CHEMBL2375494)
Affinity DataIC50:  650nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556715(CHEMBL4782344)
Affinity DataIC50:  880nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556716(CHEMBL4796964)
Affinity DataIC50:  910nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556721(CHEMBL4790746)
Affinity DataIC50:  1.01E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556719(CHEMBL4782590)
Affinity DataIC50:  1.08E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556710(CHEMBL4741257)
Affinity DataIC50:  1.23E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556706(CHEMBL4797370)
Affinity DataIC50:  1.49E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556718(CHEMBL4787771)
Affinity DataIC50:  1.52E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556699(CHEMBL4746541)
Affinity DataIC50:  1.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556705(CHEMBL4793323)
Affinity DataIC50:  1.72E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556708(CHEMBL4795327)
Affinity DataIC50:  1.76E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556722(CHEMBL4791780)
Affinity DataIC50:  1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556700(CHEMBL4761208)
Affinity DataIC50:  1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556720(CHEMBL4745132)
Affinity DataIC50:  1.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556709(CHEMBL4783011)
Affinity DataIC50:  2.37E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556703(CHEMBL4761078)
Affinity DataIC50:  2.57E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556701(CHEMBL4746014)
Affinity DataIC50:  2.63E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556702(CHEMBL4763588)
Affinity DataIC50:  2.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556704(CHEMBL4740701)
Affinity DataIC50:  3.02E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556713(CHEMBL4748854)
Affinity DataIC50:  3.29E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556714(CHEMBL4777734)
Affinity DataIC50:  3.54E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556707(CHEMBL4762863)
Affinity DataIC50:  3.87E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556723(CHEMBL240484)
Affinity DataIC50:  5.45E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556712(CHEMBL4798117)
Affinity DataIC50:  7.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50556711(CHEMBL4755423)
Affinity DataIC50:  8.13E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022147(CHEMBL3299117)
Affinity DataEC50:  646nMAssay Description:Agonist activity at GPR52 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022151(CHEMBL3299118)
Affinity DataEC50:  347nMAssay Description:Agonist activity at GPR52 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022152(CHEMBL3299018)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022153(CHEMBL3299119)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022156(CHEMBL3299120)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022157(CHEMBL3299121)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022158(CHEMBL3299122)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022159(CHEMBL3299123)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022162(CHEMBL3299124)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022164(CHEMBL3299125)
Affinity DataEC50:  646nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022165(CHEMBL3297807)
Affinity DataEC50:  209nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022166(CHEMBL3297808)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022169(CHEMBL3297809)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022170(CHEMBL3297810)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022189(CHEMBL3297811)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022190(CHEMBL3298233)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50022254(CHEMBL3298234)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50252092(CHEMBL4082756)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50252099(CHEMBL4087237)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Mus musculus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252092(CHEMBL4082756)
Affinity DataEC50:  71nMAssay Description:Agonist activity at mouse GPR52More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50252102(CHEMBL4059658)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50252136(CHEMBL4064577)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50252137(CHEMBL4074656)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50252138(CHEMBL4095110)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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