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Found 259 Enz. Inhib. hit(s) with Target = 'Gastrin-releasing peptide receptor'
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50005601(CHEMBL2369819)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408923(CHEMBL2114155)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071733(CHEMBL413196 | Compound GRP)
Affinity DataKi:  0.0400nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  0.150nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  0.150nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50066009(CHEMBL3401466)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50288252(Bombesin analogue | CHEMBL269432)
Affinity DataKi:  0.700nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071744(AcBB(7-14) | CHEMBL314375)
Affinity DataKi:  0.700nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85480((3-Ph-Pr6)His7,DAla11,DPro13,Psi13-14,Phe14-Bn(6-1...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85500(Bombesin,Phe13)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50275902(CHEMBL525577 | D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe...)
Affinity DataKi:  0.990nMAssay Description:Binding affinity to gastrin releasing peptide receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071739((S)-3-(1H-Indol-3-yl)-N-[1-(5-methoxy-pyridin-2-yl...)
Affinity DataKi:  1nMAssay Description:Antagonistic activity against cloned human Bombesin receptor bb2 labeled with [125I]- [Tyr] bombesin stably expressed in CHO cells; 0.66-1.3More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  1.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  1.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  1.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  1.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  1.52nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089280(CHEMBL437655 | JMV 1535)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  1.74nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  1.76nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089284(CHEMBL265856 | JMV 1803)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85486(DPhe6-Bn[6-14))
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85499(CAS_29451-71-6 | NSC_5489061 | Ranatensin)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85502(PG-L)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089285(CHEMBL415110 | JMV 1799)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089282((D)Phe-Gln-Trp-Ala-Val-Gly-His-Leu-Leu-NH2 | CHEMB...)
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071743((S)-3-(1H-Indol-3-yl)-N-[1-(4-methoxy-phenyl)-cycl...)
Affinity DataKi:  3.70nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089281(CHEMBL386480 | JMV 1802)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089291(CHEMBL415021 | JMV 1813)
Affinity DataKi:  5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071742((S)-N-[1-(4-Ethoxy-phenyl)-cyclohexylmethyl]-3-(1H...)
Affinity DataKi:  5.80nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85495(DPhe6-Bn(6-13)propylamide)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85498(CAS_5486808 | Litorin | NSC_5486808)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85493(DTyr6,DAla11-Bn(6-13)butylamide)
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071750((S)-3-(1H-Indol-3-yl)-2-methyl-N-[1-(4-nitro-pheny...)
Affinity DataKi:  6.40nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071741((S)-N-[1-(4-Dimethylamino-phenyl)-cyclohexylmethyl...)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089278(CHEMBL411016 | JMV 1801)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85496(DPhe6-Bn(6-13)methylester)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089279(CHEMBL406013 | JMV 1719)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071735((S)-3-(1H-Indol-3-yl)-2-methyl-2-[3-(4-nitro-pheny...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM81964(CAS_5486814 | Gastrin | NSC_5486814 | Neuromedin C)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85494(DPhe6-Bn(6-13)NH2)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM85506(CAS_125988 | NSC_125988 | Rhodei-Litorin)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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