Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with Target = 'N-methyl-D-aspartate receptor'
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089759((R)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50:  50nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of por...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50079387(1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-piperid...)
Affinity DataIC50:  83nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of por...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089759((R)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50:  213nMAssay Description:Displacement of [3H]-ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50079387(1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-piperid...)
Affinity DataIC50:  277nMAssay Description:Displacement of [3H]-ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089760((S)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50:  545nMAssay Description:Displacement of [3H]-ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089760((S)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50:  5.10E+3nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of por...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089760((S)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50:  5.10E+3nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50079387(1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-piperid...)
Affinity DataIC50:  1.13E+4nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-methyl-D-aspartate receptor(Sus scrofa)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089759((R)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50:  2.37E+4nMAssay Description:Compound was tested for inhibition of [3H]-MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed