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Found 33 Enz. Inhib. hit(s) with Target = 'Integrin alpha-2/beta-1 [T112H]'
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19053((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  15nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19066((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(3,5-d...)
Affinity DataIC50:  17nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19057((2S)-3-({[(4-aminophenyl)methyl]carbamoyl}amino)-2...)
Affinity DataIC50:  23nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19063((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(3,5-d...)
Affinity DataIC50:  29nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19065((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(3,5-d...)
Affinity DataIC50:  35nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19070((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(4-met...)
Affinity DataIC50:  36nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19064((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-{[3,5-b...)
Affinity DataIC50:  39nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19068((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-(naphth...)
Affinity DataIC50:  50nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19071((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(4-met...)
Affinity DataIC50:  70nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19066((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(3,5-d...)
Affinity DataIC50:  83nMAssay Description:The ligand was immobilized on 96-well flat microtiter in PBS buffer solution overnight, and the wells were blocked with 1% BSA in HBSS buffer solutio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19063((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(3,5-d...)
Affinity DataIC50:  89nMAssay Description:The ligand was immobilized on 96-well flat microtiter in PBS buffer solution overnight, and the wells were blocked with 1% BSA in HBSS buffer solutio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19057((2S)-3-({[(4-aminophenyl)methyl]carbamoyl}amino)-2...)
Affinity DataIC50:  102nMAssay Description:The ligand was immobilized on 96-well flat microtiter in PBS buffer solution overnight, and the wells were blocked with 1% BSA in HBSS buffer solutio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19072((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(4-nit...)
Affinity DataIC50:  105nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19058((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  107nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19061((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  108nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19074((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(4-ace...)
Affinity DataIC50:  131nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19053((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  138nMAssay Description:The ligand was immobilized on 96-well flat microtiter in PBS buffer solution overnight, and the wells were blocked with 1% BSA in HBSS buffer solutio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19073((2S)-2-{[(2S)-1-[(4-aminobenzene)sulfonyl]pyrrolid...)
Affinity DataIC50:  144nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19075((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-({4-[(p...)
Affinity DataIC50:  151nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19060((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  160nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19068((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-(naphth...)
Affinity DataIC50:  177nMAssay Description:The ligand was immobilized on 96-well flat microtiter in PBS buffer solution overnight, and the wells were blocked with 1% BSA in HBSS buffer solutio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19055((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  185nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19052((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  185nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19076((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-{[4-(2-...)
Affinity DataIC50:  236nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19069((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(4-phe...)
Affinity DataIC50:  287nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19056((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  296nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19054((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  357nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19050((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  367nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19059((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  467nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19049((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50:  660nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19051((2S)-2-{[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]f...)
Affinity DataIC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19062((2S)-2-{[(2S)-1-benzoylpyrrolidin-2-yl]formamido}-...)
Affinity DataIC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-2/beta-1 [T112H](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM19067((2S)-3-[(benzylcarbamoyl)amino]-2-{[(2S)-1-[(2,6-d...)
Affinity DataIC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:Flat bottom microtiter plates (96-well) were coated with soluble type I collagen. Unoccupied protein binding sites on the wells were blocked with bov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed