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Found 179 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 11A'
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592040(CHEMBL1989043)
Affinity DataIC50:  170nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592059(CHEMBL5175800)
Affinity DataIC50:  190nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592056(CHEMBL5185990)
Affinity DataIC50:  230nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592060(CHEMBL5180190)
Affinity DataIC50:  230nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592046(CHEMBL5185655)
Affinity DataIC50:  260nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592043(CHEMBL5206282)
Affinity DataIC50:  330nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592062(CHEMBL5200790)
Affinity DataIC50:  470nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592061(CHEMBL5208491)
Affinity DataIC50:  580nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592067(CHEMBL5173236)
Affinity DataIC50:  620nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592055(CHEMBL5200963)
Affinity DataIC50:  700nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592053(CHEMBL5184522)
Affinity DataIC50:  710nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592054(CHEMBL5182610)
Affinity DataIC50:  800nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592047(CHEMBL5171843)
Affinity DataIC50:  900nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592070(CHEMBL5194816)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592066(CHEMBL5203750)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592058(CHEMBL5180130)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592050(CHEMBL5180577)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592068(CHEMBL5190264)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592057(CHEMBL5170651)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592051(CHEMBL5180851)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592052(CHEMBL5199067)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592069(CHEMBL5177982)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592045(CHEMBL5169674)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592065(CHEMBL5190514)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592063(CHEMBL5178437)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592048(CHEMBL5207135)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592049(CHEMBL5173735)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592044(CHEMBL5200515)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592042(CHEMBL5189171)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592041(CHEMBL5192162)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50592064(CHEMBL5195298)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminus or C-terminus NLuc fused CDK11A (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM21079(1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-...)
Affinity DataKd:  1.20E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM31085(1-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluorom...)
Affinity DataKd:  1.10E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM26300(2-{3-[(7-{3-[ethyl(2-hydroxyethyl)amino]propoxy}qu...)
Affinity DataKd:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM5931(BMS-387072 | CHEMBL296468 | N-(5-{[(5-tert-butyl-1...)
Affinity DataKd:  48nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM26474(5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...)
Affinity DataKd:  1.30E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)
Affinity DataKd:  110nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKd:  260nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM13535(4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM15138(5-indazolyl pyridine 11g | 5-{5-[(2S)-2-amino-3-ph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CDC2L2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM25084(3-[2,4-diamino-6-(3-hydroxyphenyl)pteridin-7-yl]ph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CDC2L2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50355501(INCB-018424 | RUXOLITINIB | RUXOLITINIB PHOSPHATE ...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CDC2L2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM24654(4-N-(2,6-dichlorobenzene)-3-N-(piperidin-4-yl)-1H-...)
Affinity DataKd:  5.20nMAssay Description:Binding constant for CDC2L2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 11A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50128285(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmet...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CDC2L2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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