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Found 18 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-4'
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185624((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  7.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185625(CHEMBL380390 | pAM-FKF)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185645((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185646(CHEMBL207452 | Pam-YKF)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185633((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  3.15E+5nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577131(CHEMBL4855915)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577116(CHEMBL4872258)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577133(CHEMBL4870115)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50604328(CHEMBL5180795)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50604305(CHEMBL5209480)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50604324(CHEMBL5183361)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed