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Found 27 Enz. Inhib. hit(s) with Target = 'cAMP-dependent protein kinase type I-alpha regulatory subunit'
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM50011236(CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-ami...)
Affinity DataIC50:  3.60E+3nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM92674(Isoquinolinesulfonamide, CKI-7)
Affinity DataIC50:  5.50E+5nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM92673(Isoquinolinesulfonamide, CKI-6)
Affinity DataIC50: >1.00E+6nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81290(MLS001148197 | N6,2'-O-DIBUTYRYLADENOSINE-3...)
Affinity DataEC50:  4.48E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81291(8-(4-Chlorophenylthio)adenosine 3',5'-cycl...)
Affinity DataEC50:  32.7nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81292(8-Bromoadenosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  34.4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM66980(Bucladesine sodium salt | MLS002154012 | SMR001233...)
Affinity DataEC50:  6.70E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81290(MLS001148197 | N6,2'-O-DIBUTYRYLADENOSINE-3...)
Affinity DataEC50:  1.23E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81294(3-[(2,4-dichlorobenzyl)sulfanyl]-2-thiophenecarbox...)
Affinity DataEC50: >1.14E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81295(4-{(E)-[4-(dimethylamino)-1-naphthyl]diazenyl}benz...)
Affinity DataEC50: >1.14E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81287(6-(6-aminopurin-9-yl)-2-ethoxy-2-oxidanylidene-4a,...)
Affinity DataEC50:  2.68E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81288(8-Bromoguanosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  7.83E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM51788(5-[(2E)-2-(8-oxidanylidenequinolin-5-ylidene)hydra...)
Affinity DataEC50: >1.14E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81289(Adenosine 3',5'-cyclic monophosphate sodiu...)
Affinity DataEC50:  68.0nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81290(MLS001148197 | N6,2'-O-DIBUTYRYLADENOSINE-3...)
Affinity DataEC50:  4.48E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81291(8-(4-Chlorophenylthio)adenosine 3',5'-cycl...)
Affinity DataEC50:  32.7nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81292(8-Bromoadenosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  34.4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM66980(Bucladesine sodium salt | MLS002154012 | SMR001233...)
Affinity DataEC50:  6.70E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81290(MLS001148197 | N6,2'-O-DIBUTYRYLADENOSINE-3...)
Affinity DataEC50:  1.23E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Homo sapiens (Human))
University Of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.30nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [R241A](Homo sapiens (Human))
University Of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  6.72nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [K242A](Homo sapiens (Human))
University Of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.32nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [R243A](Homo sapiens (Human))
University Of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.29nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81289(Adenosine 3',5'-cyclic monophosphate sodiu...)
Affinity DataEC50:  68.0nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [K244A](Homo sapiens (Human))
University Of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.71nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81287(6-(6-aminopurin-9-yl)-2-ethoxy-2-oxidanylidene-4a,...)
Affinity DataEC50:  2.68E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM81288(8-Bromoguanosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  7.83E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay