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Found 5 Enz. Inhib. hit(s) with Target = 'Signal transducer and activator of transcription 3 [127-722]'
TargetSignal transducer and activator of transcription 3 [127-722](Mus musculus (mouse))
University Of Michigan At Ann Arbor

LigandPNGBDBM28130(4-[(2S)-2-{[(3S)-1-({[(1S)-1-(benzylcarbamoyl)-3-c...)
Affinity DataKi:  190nM ΔG°:  -38.0kJ/molepH: 7.5 T: 2°CAssay Description:The assay was based on the fluorescence polarization of the unbound small binding partner will be low, and its binding to a larger binding partner wi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3 [127-722](Mus musculus (mouse))
University Of Michigan At Ann Arbor

LigandPNGBDBM28128(4-[(2S)-2-{[(2S)-1-[(2S)-2-{[(1S)-1-(benzylcarbamo...)
Affinity DataKi:  350nM ΔG°:  -36.5kJ/molepH: 7.5 T: 2°CAssay Description:The assay was based on the fluorescence polarization of the unbound small binding partner will be low, and its binding to a larger binding partner wi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3 [127-722](Mus musculus (mouse))
University Of Michigan At Ann Arbor

LigandPNGBDBM28129(4-[(2S)-2-{[(3S)-1-({[(1S)-1-(benzylcarbamoyl)-3-c...)
Affinity DataKi:  3.13E+3nM ΔG°:  -31.1kJ/molepH: 7.5 T: 2°CAssay Description:The assay was based on the fluorescence polarization of the unbound small binding partner will be low, and its binding to a larger binding partner wi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3 [127-722](Mus musculus (mouse))
University Of Michigan At Ann Arbor

LigandPNGBDBM20246(4-[(2S)-2-{[(1S)-1-{[(6S,9S,12S)-12-{[(1S)-1-carba...)
Affinity DataKi:  7.30E+3nM ΔG°:  -29.0kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization (FP) binding assay is utilizing the intrinsic property of the fluorescent probe, which will have low polarization value whe...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3 [127-722](Mus musculus (mouse))
University Of Michigan At Ann Arbor

LigandPNGBDBM20244(4-[(2S)-2-{[(1S)-1-{[(1S)-5-amino-1-{[(1S,2R)-1-{[...)
Affinity DataKi:  2.59E+4nM ΔG°:  -25.9kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization (FP) binding assay is utilizing the intrinsic property of the fluorescent probe, which will have low polarization value whe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed