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Found 24 Enz. Inhib. hit(s) with Target = 'Tubulin--tyrosine ligase'
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM18129((2S)-2-amino-3-(4-hydroxyphenyl)propanoic acid | L...)
Affinity DataKi:  2.50E+4nM ΔG°:  -27.3kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36556(3-Azidotyrosine)
Affinity DataKi:  2.00E+5nM ΔG°:  -22.0kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36555(3-Aminotyrosine)
Affinity DataKi:  2.00E+5nM ΔG°:  -22.0kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36557(3-Formyltyrosine)
Affinity DataKi:  3.00E+5nM ΔG°:  -20.9kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36554(3-Nitrotyrosine)
Affinity DataKi:  4.00E+5nM ΔG°:  -20.2kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM36558(4-Aminophenylalanine)
Affinity DataKi: >4.00E+6nM ΔG°: >-14.2kJ/molepH: 6.8 T: 2°CAssay Description:Inhibition of [3H]-L-tyrosine incorporation into tubulin by enzyme tubulin tyrosine ligase (TTL).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293291(6alpha,15(S)-dihydroxy-23-oxo-labd-8(22),13(14),17...)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293292(6alpha,15(S),23-trihydroxy-labd-8(22),13(14),17-tr...)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293293(6alpha,8alpha-dihydroxy-23-oxo-labd-13(14),17-dien...)
Affinity DataKd:  810nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293294(6alpha,8alpha,15(S)-trihydroxy-23-oxo-labd-13(14),...)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293295(6alpha,8alpha,15(S)-trihydroxy-23-carbossimethylla...)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293296(6alpha,8alpha-dihydroxy-23-carbossi-labd-13(14),17...)
Affinity DataKd:  7nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293297(6alpha,8alpha,15(S)-trihydroxy-23-carbossi-labd-13...)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293298(6alpha,8alpha,23-trihydroxy-labd-13(14),17-dien-16...)
Affinity DataKd:  72nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293299(6alpha,8alpha,15(S),23-tetrahydroxy-labd-13(14),17...)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293300(8alpha-hydroxy,23alpha-O-ethyl-23,6alpha-epoxy-lab...)
Affinity DataKd:  73nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293301(8alpha,15(S)-dihydroxy,23alpha-O-ethyl-23,6alpha-e...)
Affinity DataKd:  960nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293302(8alpha,15(S),23alpha-trihydroxy-23,6alpha-epoxy-la...)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293289(6alpha,8alpha-dihydroxy-23-carbossi-labd-13(14),15...)
Affinity DataKd:  93nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293288(6alpha,8alpha-dihydroxy-23-oxo-13(14),15,17-trien-...)
Affinity DataKd:  200nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293287(8alpha-hydroxylabd-13(14),15,17-trien-6alpha,23-16...)
Affinity DataKd:  150nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293286(8alpha-23-dihydroxy-23,6alpha-epoxy-labd-13(14),15...)
Affinity DataKd:  480nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293285(23,6alpha-epoxy-labd-8,13(14),17-trien-16(R),19-ol...)
Affinity DataKd:  8.70E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Binghamton University

LigandPNGBDBM50293290(6alpha,8alpha,23-trihydroxy-labd-13(14),15,17-trie...)
Affinity DataKd:  110nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed