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Found 21 Enz. Inhib. hit(s) with Target = 'Uridine-cytidine kinase 2'
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522195(CHEMBL1592234)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using uridine, phosphoenolpyruvate, N...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522195(CHEMBL1592234)
Affinity DataKi:  3.50E+3nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using phosphoenolpyruvate, NADH and v...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522193(CHEMBL4553820)
Affinity DataKi:  1.20E+4nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using uridine, phosphoenolpyruvate, N...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522193(CHEMBL4553820)
Affinity DataKi:  1.30E+4nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using phosphoenolpyruvate, NADH and v...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522198(CHEMBL4434988)
Affinity DataKi:  3.10E+4nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using uridine, phosphoenolpyruvate, N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522198(CHEMBL4434988)
Affinity DataKi:  5.00E+4nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using phosphoenolpyruvate, NADH and v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522195(CHEMBL1592234)
Affinity DataIC50:  3.00E+3nMAssay Description:Non-competitive inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells using phosphoenolpyruvate, NADH, urid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522195(CHEMBL1592234)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522201(CHEMBL4588628)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522193(CHEMBL4553820)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522197(CHEMBL4575982)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522193(CHEMBL4553820)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522198(CHEMBL4434988)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522196(CHEMBL4589970)
Affinity DataIC50:  2.68E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522198(CHEMBL4434988)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522195(CHEMBL1592234)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522194(CHEMBL1564286)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522199(CHEMBL4564613)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522200(CHEMBL1514618)
Affinity DataIC50:  1.38E+5nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM50522202(CHEMBL4457001)
Affinity DataIC50:  1.66E+5nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUridine-cytidine kinase 2(Homo sapiens)
Stanford University

Curated by ChEMBL
LigandPNGBDBM48877(3-[({[2-(4-fluorophenyl)-5H-chromeno[2,3-d]pyrimid...)
Affinity DataIC50:  1.66E+5nMAssay Description:Inhibition of C-terminally His6-tagged human UCK2 expressed in Escherichia coli BL21(DE3) cells incubated for 15 mins before ATP addition and measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed